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Sigma-1 receptor antagonist 2

Catalog No.GC38039

Sigma-1 receptor antagonist 2 is a potent and selective sigma 1 receptor (σ1 R) antagonist with Kis of 3.88 and 1288 nM for σ1 and σ2 receptor, respectively.

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Sigma-1 receptor antagonist 2 Chemical Structure

Cas No.: 1639220-15-7

Size Price Stock Qty
10mM (in 1mL DMSO)
$297.00
In stock
1mg
$202.00
In stock
5mg
$270.00
In stock
10mg
$450.00
In stock

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Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents Related Products

Sigma-1 receptor antagonist 2 is a potent and selective sigma 1 receptor (σ1 R) antagonist with Kis of 3.88 and 1288 nM for σ1 and σ2 receptor, respectively[1].

[1]. Lan Y, et al. Synthesis and biological evaluation of novel sigma-1 receptor antagonists based on pyrimidine scaffold as agents for treating neuropathic pain. J Med Chem. 2014 Dec 26;57(24):10404-23.

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