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Home >> Signaling Pathways >> GPCR/G protein >> CaSR

CaSR

CASR (calcium sensing receptor) is a G-protein couple receptor which regulates the calcium homeostasis and involved in proliferation, differentiation and other hormonal secretion.

Products for  CaSR

  1. Cat.No. Product Name Information
  2. GC64905 (Rac)-Upacicalcet (Rac)-Upacicalcet is the racemate of Upacicalcet. (Rac)-Upacicalcet Chemical Structure
  3. GC50365 AC 265347 Biased allosteric modulator of calcium-sensing receptor (CaSR) AC 265347 Chemical Structure
  4. GC17244 Calcium-Sensing Receptor Antagonists I Calcium-Sensing Receptor Antagonists I Chemical Structure
  5. GC17697 Calhex 231 hydrochloride

    negative allosteric modulator of Ca2+-sensing receptor (CaSR)

     Calhex 231 hydrochloride Chemical Structure
  6. GC12620 Calindol (hydrochloride) activator of the calcium-sensing receptor (CaSR) Calindol (hydrochloride) Chemical Structure
  7. GC13518 Cinacalcet Cinacalcet Chemical Structure
  8. GC16708 Cinacalcet HCl

    AMG 073, KRN 1493, Mimpara

     Cinacalcet HCl (AMG-073 hydrochloride) is an orally active, allosteric agonist of Ca receptor (CaR), used for cardiovascular disease treatment. Cinacalcet HCl Chemical Structure
  9. GC63745 Cinacalcet-D3

    AMG 073-D3

     Cinacalcet-D3 Chemical Structure
  10. GC38148 Etelcalcetide Etelcalcetide (AMG 416) is a synthetic peptide as an activator of the calcium sensing receptor (CaSR). Etelcalcetide Chemical Structure
  11. GC38147 Etelcalcetide hydrochloride

    KAI 4169, Velcalcetide

     A peptide agonist of CaSR Etelcalcetide hydrochloride Chemical Structure
  12. GC30389 Evocalcet (KHK7580)

    KHK7580, MT-4580

     Evocalcet (KHK7580) has an activating effect on calcium sensing receptor (CaSR) extracted from patent WO 2017061621 A1, compound A. Evocalcet (KHK7580) Chemical Structure
  13. GC69193 GSK3004774

    GSK3004774 is an effective, non-absorbable CaSR agonist with pEC50 values of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR respectively, and an EC50 value of 50 nM for human CaSR.

     GSK3004774 Chemical Structure
  14. GN10419 Ligustroflavone Ligustroflavone Chemical Structure
  15. GC16943 NPS-2143 NPS-2143 is a calcification drug that acts as an antagonist of the calcium-sensing receptor (CaSR) and consequently stimulates the release of parathyroid hormone. NPS-2143 Chemical Structure
  16. GC12240 NPS-2143 hydrochloride

    SB-262470A

     An orally-active CaSR antagonist NPS-2143 hydrochloride Chemical Structure
  17. GC17700 R 568 hydrochloride

    KRN 568, NPS R-568, Tecalcet

     R 568 hydrochloride (R 568 Hydrochloride), an orally active calcimimetic compound, allosterically and positively modulates the calcium-sensing receptor (CaSR). R 568 hydrochloride Chemical Structure
  18. GC30095 SB-423562 SB-423562 is a short-acting calcium-sensing receptor (CaR) antagonist. SB-423562 Chemical Structure
  19. GC12442 Strontium chloride Calcium sensing receptor (CaSR) agonist Strontium chloride Chemical Structure
  20. GC11819 Strontium Ranelate

    S12911, S12911-2

     Calcium Channel activator Strontium Ranelate Chemical Structure
  21. GC64923 Upacicalcet sodium Upacicalcet sodium is an intravenous calcimimetic agent. Upacicalcet sodium Chemical Structure

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