RS 127445 hydrochloride |
| Catalog No.GC50033 |
High affinity and selective 5-HT2B antagonist
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 199864-86-3
Sample solution is provided at 25 µL, 10mM.
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High affinity 5-HT2B receptor antagonist (pKi = 9.5). Displays 1000-fold selectivity for 5-HT2B with good bioavailability.
Bonhaus et al (1999) RS-127445: a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist. Br.J.Pharmacol. 127 1075 PMID:10455251 |Callebert et al (2006) Evidence for a control of plasma serotonin levels by 5-Hydroxytryptamine2B receptors in mice. J.Pharmacol.Exp.Ther. 317 724 PMID:16461587
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