P450
Products for P450
- Cat.No. Product Name Information
- GC10136 Tienilic Acid Suicide substrate of CYP 2C9
- GC15445 TMS cytochrome P450 1B1 inhibitor
- GC13362 TOK-001 TOK-001 (TOK-001) is a multifunctional antiandrogen and CYP17 inhibitor (IC50=47 nM) in castration resistant prostate cancer (CRPC).
- GC45582 trans-ε-Viniferin ε-Viniferin, the dimer of Resveratrol and isolated from Vitis vinifera, displays a potent inhibitory for all the CYP activities, with Ki values from 0.5-20 μM.
- GC49212 trans-carboxy Glimepiride A metabolite of glimepiride
- GC52060 Trimipramine N-oxide Trimipramine N-oxide is an active metabolite of the tricyclic antidepressant trimipramine.
- GC17112 Uniconazole cytochrome P450 707As inhibitor
- GC31791 Veledimex (INXN-1001) Veledimex (INXN-1001) (INXN-1001), a synthetic analog of the insect molting hormone ecdysone, is an orally active activator ligand for a proprietary gene therapy promoter system.
- GC33870 Veledimex racemate (RG-115932 racemate) Veledimex racemate (RG-115932 racemate) (INXN-1001 racemate) is the racemate of veledimex.
- GC30705 Veledimex S enantiomer (INXN-1001 S enantiome) Veledimex S enantiomer (INXN-1001 S enantiomer) is the S enantiomer of veledimex. Veledimex is an oral activator ligand for a proprietary gene therapy promoter system, and a moderate inhibitor of and substrate for CYP3A4/5.
- GC61811 Verapamil Verapamil ((±)-Verapamil) is a calcium channel blocker and a potent and orally active first-generation P-glycoprotein (P-gp) inhibitor.
- GC45151 Voriconazole N-oxide Voriconazole N-oxide is a major metabolite of the triazole antifungal voriconazole.
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GC15056
β-Nicotyrine
cytochrome P450 (CYP) isoforms, CYP2A6 and CYP2A13 inhibitor