Search Site
  • 0
    My Cart

    Click Here to Find How Many Items You Have Added:)

    image loader

    Adding item(s) to cart......

Home >> Signaling Pathways >> Proteases >> Drug Metabolite

Drug Metabolite

Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.

Targets for  Drug Metabolite

Products for  Drug Metabolite

  1. Cat.No. Product Name Information
  2. GC39373 Desmethyl ferroquine Desmethyl ferroquine (SSR97213) is the active and major metabolite of Ferroquine. Desmethyl ferroquine Chemical Structure
  3. GC49202 Desmethyl Mirtazapine (hydrochloride) A metabolite of mirtazapine Desmethyl Mirtazapine (hydrochloride) Chemical Structure
  4. GC49100 Desmethyl Ofloxacin (hydrochloride) A metabolite of ofloxacin Desmethyl Ofloxacin (hydrochloride) Chemical Structure
  5. GC49409 Desmethyl Ranolazine A metabolite of ranolazine Desmethyl Ranolazine Chemical Structure
  6. GC49870 Desmethyl Sibutramine (hydrochloride) An active metabolite of sibutramine Desmethyl Sibutramine (hydrochloride) Chemical Structure
  7. GC43422 Desmethyldoxepin (hydrochloride) Desmethyldoxepin (hydrochloride) is the major metabolite of Doxepin. Desmethyldoxepin (hydrochloride) Chemical Structure
  8. GC43423 Desmethylene Paroxetine (hydrochloride) Paroxetine is a potent, selective serotonin reuptake inhibitor (Ki = 0.72 nM) that has been used in cases of depression and anxiety disorder. Desmethylene Paroxetine (hydrochloride) Chemical Structure
  9. GC60132 Desmethylnortriptyline Desmethylnortriptyline is a metabolite of Nortriptyline. Desmethylnortriptyline Chemical Structure
  10. GC43444 Diclofenac Acyl-β-D-Glucuronide Diclofenac acyl-β-D-glucuronide is an active metabolite of diclofenac and the predominant metabolite in rat. Diclofenac Acyl-β-D-Glucuronide Chemical Structure
  11. GC49842 Digoxigenin Bisdigitoxoside A Na+/K+-ATPase inhibitor Digoxigenin Bisdigitoxoside Chemical Structure
  12. GC18455 Digoxigenin Monodigitoxoside Digoxigenin monodigitoxoside is a Na+/K+-ATPase inhibitor and cardiac glycoside metabolite of digoxin . Digoxigenin Monodigitoxoside Chemical Structure
  13. GC40143 Dihydrotetrabenazine Dihydrotetrabenazine is an active metabolite of the vesicular monoamine transporter 2 (VMAT2) inhibitor tetrabenazine that is generated by hepatic carbonyl reductases. Dihydrotetrabenazine Chemical Structure
  14. GC64759 Dimethadione Dimethadione is the primary metabolite of trimethadione. Dimethadione Chemical Structure
  15. GC61864 DL-Laudanosine DL-Laudanosine, an Atracurium and Cisatracurium metabolite, crosses the blood–brain barrier and may cause excitement and seizure activity. DL-Laudanosine Chemical Structure
  16. GC52368 DL-Sulforaphane Glutathione A metabolite of sulforaphane DL-Sulforaphane Glutathione Chemical Structure
  17. GC43493 DL-Sulforaphane N-acetyl-L-cysteine Nrf2 activation of the antioxidant response element (ARE) is central to cytoprotective gene expression against oxidative and/or electrophilic stress. DL-Sulforaphane N-acetyl-L-cysteine Chemical Structure
  18. GC52052 Dofetilide N-oxide Dofetilide N-oxide Chemical Structure
  19. GC49288 Dolutegravir M1 A metabolite of dolutegravir Dolutegravir M1 Chemical Structure
  20. GC49289 Dolutegravir O-β-D-Glucuronide A metabolite of dolutegravir Dolutegravir O-β-D-Glucuronide Chemical Structure
  21. GC40018 Donepezil N-oxide Donepezil N-oxide is an active metabolite of the acetylcholinesterase inhibitor donepezil. Donepezil N-oxide Chemical Structure
  22. GC18439 Doxorubicinone A metabolite of doxorubicin Doxorubicinone Chemical Structure
  23. GC63389 DP-1 DP-1, a degradation product of SDC-TRAP-0063, is a fragment of Ganetespib. DP-1 Chemical Structure
  24. GC33571 Duloxetine metabolite Para-Naphthol Duloxetine (Para-Naphthol duloxetine) Para-Naphthol Duloxetine is a metabolite of Duloxetine, which is a serotonin-norepinephrine reuptake inhibitor (SNRI). Duloxetine metabolite Para-Naphthol Duloxetine (Para-Naphthol duloxetine) Chemical Structure
  25. GC65956 Edoxaban M4 Edoxaban M4, an active metabolite of Edoxaban, shows reproducible, but concentration-dependent matrix effects. Edoxaban (DU-176) is a selective, potent and orally active factor Xa (FXa) inhibitor . Edoxaban M4 Chemical Structure
  26. GC35990 Endoxifen hydrochloride Endoxifen hydrochloride is a key active metabolite of Tamoxifen (TAM) with higher affinity and specificity to estrogen receptor that also inhibits aromatase activity. Endoxifen hydrochloride has the potential for breast cancer study. Endoxifen hydrochloride Chemical Structure
  27. GC16292 Equol non-steroidal estrogen Equol Chemical Structure
  28. GC12685 Ercalcitriol A potent agonist of the vitamin D receptor Ercalcitriol Chemical Structure
  29. GC45449 Erythromycylamine   Erythromycylamine Chemical Structure
  30. GC52035 Esmolol Acid (hydrochloride) An active metabolite of esmolol Esmolol Acid (hydrochloride) Chemical Structure
  31. GC48979 Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate) A substrate of multidrug resistance protein 2 Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate) Chemical Structure
  32. GC47320 Ethynyl Estradiol 3-β-D-Glucuronide (hydrate) A metabolite of ethynyl estradiol Ethynyl Estradiol 3-β-D-Glucuronide (hydrate) Chemical Structure
  33. GC38779 Etilevodopa Etilevodopa (L-Dopa ethyl ester), an ethyl-ester prodrug of Levodopa, is rapidly hydrolyzed to Levodopa and ethanol by nonspecific esterases in the gastrointestinal tract. Etilevodopa Chemical Structure
  34. GC39757 Etilevodopa hydrochloride Etilevodopa (L-Dopa ethyl ester) hydrochloride, an ethyl-ester prodrug of Levodopa, is rapidly hydrolyzed to Levodopa and ethanol by nonspecific esterases in the gastrointestinal tract. Etilevodopa hydrochloride Chemical Structure
  35. GC49156 Etodolac Acyl Glucuronide A phase II metabolite of etodolac Etodolac Acyl Glucuronide Chemical Structure
  36. GC43646 Ezetimibe Hydroxy Glucuronide Ezetimibe hydroxy glucuronide is a minor phase II glucuronide metabolite of ezetimibe . Ezetimibe Hydroxy Glucuronide Chemical Structure
  37. GC60831 Ezetimibe phenoxy glucuronide Ezetimibe phenoxy glucuronide (Ezetimibe glucuronide) is the active metabolite of Ezetimibe. Ezetimibe phenoxy glucuronide Chemical Structure
  38. GC40190 Febuxostat Acyl Glucuronide Febuxostat acyl glucuronide is a metabolite of the xanthine oxidoreductase inhibitor febuxostat. Febuxostat Acyl Glucuronide Chemical Structure
  39. GC66449 Ferulic acid 4-O-sulfate Ferulic acid 4-O-sulfate (Ferulic acid 4-sulfate) is a metabolite of Ferulic acid (HY-N0060). Ferulic acid 4-O-sulfate relaxes arteries and lowers blood pressure in mice. Ferulic acid 4-O-sulfate Chemical Structure
  40. GC68387 FGN849 FGN849 Chemical Structure
  41. GC43675 Florfenicol amine (hydrochloride) Florfenicol amine is a major metabolite of the antibiotic florfenicol, a fluorinated derivative of chloramphenicol that is commonly used in veterinary medicine. Florfenicol amine (hydrochloride) Chemical Structure
  42. GC36058 Flumazenil acid Flumazenil acid is a metabolite of Flumazenil. Flumazenil acid Chemical Structure
  43. GC43697 Formoterol O-β-D-Glucuronide Formoterol O-β-D-glucuronide is a metabolite of formoterol . Formoterol O-β-D-Glucuronide Chemical Structure
  44. GC62278 FTISADTSK acetate FTISADTSK acetate is an endogenous stable signature peptide from Trastuzumab monitored by selected reaction monitoring (SRM). FTISADTSK acetate Chemical Structure
  45. GC43743 Gemfibrozil 1-O-β-Glucuronide Gemfibrozil 1-O-β-glucuronide is a major metabolite of gemfibrozil that is formed when gemfibrozil undergoes glucuronidation by UDP-glucuronosyltransferase (UGT) 2B7. Gemfibrozil 1-O-β-Glucuronide Chemical Structure
  46. GC48720 Griseofulvic Acid A metabolite of griseofulvin Griseofulvic Acid Chemical Structure
  47. GC60181 GS-704277

    An intermediate alanine metabolite of remdesivir

     GS-704277 Chemical Structure
  48. GC49855 Harmalol (hydrochloride hydrate) A β-carboline alkaloid and an active metabolite of harmaline Harmalol (hydrochloride hydrate) Chemical Structure
  49. GC62152 Homovanillyl alcohol Homovanillyl alcohol is a biological metabolite of Hydroxytyrosol. Homovanillyl alcohol Chemical Structure
  50. GC49130 Hydroxy Celecoxib An inactive metabolite of celecoxib Hydroxy Celecoxib Chemical Structure
  51. GC43878 Hydroxy Dimetridazole Hydroxy Dimetridazole (Hydroxy dimetridazole) is a hydroxy metabolite of Dimetridazole. Hydroxy Dimetridazole Chemical Structure
  52. GC43879 Hydroxy Ebastine Hydroxy Ebastine is an ebastine metabolite. Hydroxy Ebastine Chemical Structure
  53. GC33438 Hydroxy Itraconazole Hydroxy Itraconazole (Itraconazole metabolite Hydroxy Itraconazole; R-63373) is an active metabolite of Itraconazole (ITZ), which is a triazole antifungal agent. Hydroxy Itraconazole Chemical Structure
  54. GC49282 Hydroxy Lenalidomide A metabolite of lenalidomide Hydroxy Lenalidomide Chemical Structure
  55. GC64511 Hydroxy ritonavir Hydroxy ritonavir is a metabolite of Ritonavir. Hydroxy ritonavir Chemical Structure
  56. GC43881 Hydroxy Varenicline A metabolite of varenicline Hydroxy Varenicline Chemical Structure
  57. GC49250 Hydroxydehydro Nifedipine Carboxylate A metabolite of nifedipine Hydroxydehydro Nifedipine Carboxylate Chemical Structure
  58. GC60920 Hydroxyhexamide Hydroxyhexamide is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agents. Hydroxyhexamide Chemical Structure
  59. GC32482 Hydroxyhexamide ((±)-Hydroxyhexamid) Hydroxyhexamide ((±)-Hydroxyhexamid) Chemical Structure
  60. GC49559 Hydroxymethyl Tolperisone (hydrochloride) A metabolite of tolperisone Hydroxymethyl Tolperisone (hydrochloride) Chemical Structure
  61. GC49832 Hydroxymetronidazole Hydroxymetronidazole (Metronidazole-OH) is a metabolite of Metronidazole belonging to the class of nitroimidazoles. Hydroxymetronidazole Chemical Structure
  62. GC40191 Ibuprofen Carboxylic Acid Ibuprofen carboxylic acid is a major metabolite of ibuprofen. Ibuprofen Carboxylic Acid Chemical Structure
  63. GC43895 Iloperidone metabolite P88 Iloperidone metabolite P88 (P88; Hydroxy Iloperidone) is a metabolite of Iloperidone, which is an atypical antipsychotic. Iloperidone metabolite P88 Chemical Structure
  64. GC43896 Iloperidone metabolite P95 Iloperidone metabolite P95 is a metabolite of the atypical antipsychotic iloperidone. Iloperidone metabolite P95 Chemical Structure
  65. GC49218 Imidafenacin Metabolite M4 A metabolite of imidafenacin Imidafenacin Metabolite M4 Chemical Structure
  66. GC64720 Imipramine N-oxide Imipramine N-oxide is the metabolite of Imipramine. Imipramine N-oxide Chemical Structure
  67. GC36304 IMR-1A IMR-1A, a acid metabolite of IMR-1, is a Notch inhibitor with an IC50 of 0.5 μM. IMR-1A has a 50-fold increase in potency with respect to IMR-1. IMR-1 can metabolize in vivo to IMR-1A. IMR-1A Chemical Structure
  68. GC49698 Indomethacin Acyl Glucuronide A metabolite of indomethacin Indomethacin Acyl Glucuronide Chemical Structure
  69. GC39119 Isonicotinic acid Isonicotinic acid is a metabolite of Isoniazid. Isonicotinic acid Chemical Structure
  70. GC33578 Ivabradine metabolite N-Demethyl Ivabradine hydrochloride N-Demethyl Ivabradine Hcl is a metabolite of Ivabradine, which is a specific inhibitor of the funny channel. Ivabradine metabolite N-Demethyl Ivabradine hydrochloride Chemical Structure
  71. GC63028 IYPTNGYTR acetate IYPTNGYTR acetate, a deamidation-sensitive signature peptide, is a deamidation product of Trastuzumab. IYPTNGYTR acetate Chemical Structure
  72. GC49538 Lamotrigine N2-oxide A metabolite of lamotrigine Lamotrigine N2-oxide Chemical Structure
  73. GC44033 Lansoprazole sulfone Lansoprazole sulfone is a phase I metabolite of lansoprazole. Lansoprazole sulfone Chemical Structure
  74. GC40099 Leukotriene D4 MaxSpec® Standard Leukotriene D4 MaxSpec® Standard is a potent bronchoconstrictor. Leukotriene D4 MaxSpec® Standard Chemical Structure
  75. GC40144 Levofloxacin N-oxide Levofloxacin N-oxide is an inactive metabolite of the antibiotic levofloxacin. Levofloxacin N-oxide Chemical Structure
  76. GC52074 Loratadine N-oxide Loratadine n-oxide is a metabolite of Loratadine. Loratadine N-oxide Chemical Structure
  77. GC41177 Lurasidone metabolite 14283 Lurasidone metabolite 14283 is an active metabolite of the atypical antipsychotic lurasidone . Lurasidone metabolite 14283 Chemical Structure
  78. GC34413 Lurasidone Metabolite 14283 D8 Lurasidone Metabolite 14283 D8 Chemical Structure
  79. GC33672 Lurasidone Metabolite 14283 hydrochloride Lurasidone Metabolite 14283 hydrochloride is a major active metabolite of Lurasidone. Lurasidone Metabolite 14283 hydrochloride Chemical Structure
  80. GC33564 Lurasidone metabolite 14326 An active metabolite of lurasidone Lurasidone metabolite 14326 Chemical Structure
  81. GC34411 Lurasidone Metabolite 14326 D8 Lurasidone Metabolite 14326 D8 is the deuterium labeled Lurasidone Metabolite 14326, which is a metabolite of Lurasidone. Lurasidone Metabolite 14326 D8 Chemical Structure
  82. GC34412 Lurasidone metabolite 14326 hydrochloride Lurasidone metabolite 14326 (hydrochloride) is an active metabolite of the atypical antipsychotic Lurasidone. Lurasidone metabolite 14326 hydrochloride Chemical Structure
  83. GC61037 Mebeverine acid Mebeverine acid (Mebeverine metabolite Mebeverine acid) is a secondary metabolite of Mebeverine. Mebeverine acid Chemical Structure
  84. GC39404 Mebeverine alcohol Mebeverine alcohol is a metabolite of Mebeverine, which is a musculotropic antispasmodic drug. Mebeverine alcohol Chemical Structure
  85. GC49755 Meclizine N-oxide A metabolite of meclizine Meclizine N-oxide Chemical Structure
  86. GC38660 Megestrol Megestrol is a synthetic progestin and used for the treatment of anorexia, cachexia, or an unexplained significant weight loss in patients with an acquired immunodeficiency syndrome diagnosis. Megestrol Chemical Structure
  87. GC45508 MEGX (hydrochloride)   MEGX (hydrochloride) Chemical Structure
  88. GC36589 Methotrexate metabolite Methotrexate metabolite (DAMPA), the active metabolite of Methotrexate. Methotrexate metabolite Chemical Structure
  89. GC49241 Methyl Diethyldithiocarbamate An active metabolite of disulfiram Methyl Diethyldithiocarbamate Chemical Structure
  90. GC49185 Mirtazapine N-oxide A metabolite of mirtazapine Mirtazapine N-oxide Chemical Structure
  91. GC32535 Modecainide (BMY 40327) Modecainide (BMY 40327) is a major metabolite of Encainide, which is an antiarrhythmic agent. Modecainide (BMY 40327) Chemical Structure
  92. GC34408 Monohydroxy Netupitant D6 Monohydroxy Netupitant D6 is the deuterium labeled Monohydroxy Netupitant, which is a metabolite of Netupitant. Monohydroxy Netupitant D6 Chemical Structure
  93. GC44246 Moxifloxacin N-Sulfate (sodium salt) Moxifloxacin N-sulfate is a metabolite of moxifloxacin. Moxifloxacin N-Sulfate (sodium salt) Chemical Structure
  94. GC41325 Mycophenolic Acid β-D-Glucuronide Mycophenolic Acid β-D-Glucuronide is a metabolite of the immunosuppressant mycophenolic acid (MPA). Mycophenolic Acid β-D-Glucuronide shows anti-tumor activity and can be used in adenocarcinoma research. Mycophenolic Acid β-D-Glucuronide Chemical Structure
  95. GC44294 N-acetyl Dapsone N-acetyl Dapsone is a metabolite of dapsone, an anti-inflammatory and antibacterial compound that is widely used in the treatment of leprosy, malaria, acne, and various immune disorders. N-acetyl Dapsone Chemical Structure
  96. GC47735 N-acetyl Desethylchloroquine-d4 An internal standard for the quantification of N-acetyl desethylchloroquine N-acetyl Desethylchloroquine-d4 Chemical Structure
  97. GC49256 N-acetyl Lenalidomide A metabolite of lenalidomide N-acetyl Lenalidomide Chemical Structure
  98. GC63337 N-Acetyl Norgestimate-d6 N-Acetyl Norgestimate-d6 Chemical Structure
  99. GC44299 N-Acetyl-4-benzoquinone imine N-Acetyl-4-benzoquinone imine is the toxic metabolite of Acetaminophen. N-Acetyl-4-benzoquinone imine Chemical Structure
  100. GC40298 N-acetyl-5-Aminosalicylic Acid N-acetyl-5-Aminosalicylic acid is a metabolite of the anti-inflammatory agent 5-aminosalicylic acid and its prodrug form, sulfasalazine. N-acetyl-5-Aminosalicylic Acid Chemical Structure
  101. GC44304 N-Acetyl-S-allyl-L-cysteine L-Deoxyalliin, also known as S-allyl-L-cysteine, is a water soluble organosulfur compound derived from garlic that has neuroprotective and antioxidative activities. N-Acetyl-S-allyl-L-cysteine Chemical Structure

Items 201 to 300 of 451 total

per page
  2. 1
  3. 2
  4. 3
  5. 4
  6. 5

Set Descending Direction