PF-02575799 |
| Catalog No.GC31522 |
PF-02575799 is a microsomal triglyceride transfer protein (MTP) inhibitor with an IC50 of 0.77±0.29 nM.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 863491-70-7
Sample solution is provided at 25 µL, 10mM.
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PF-02575799 is a microsomal triglyceride transfer protein (MTP) inhibitor with an IC50 of 0.77±0.29 nM.
PF-02575799 is compound 13 from the reference[1].
PF-02575799 produces appreciable triglyceride effects at its minimally effective dose (10 mg/kg). PF-02575799 significant increase alanine transaminase at 100 mg/kg[1].
[1]. Robinson RP, et al. Discovery of microsomal triglyceride transfer protein (MTP) inhibitors with potential for decreased active metabolite load compared to dirlotapide. Bioorg Med Chem Lett. 2011 Jul 15;21(14):4150-4.
Average Rating: 5 (Based on Reviews and 13 reference(s) in Google Scholar.)
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