Neuroscience
Neuroscience
Neurons communicate with each other, effector organs and sensory organs through the neurotransmitter – receptor pathway at synapses. Neurotransmitters can be divided into 4 major groups: 1. Amino acids (glumate, aspartate, serine, glycine and GABA); 2. Monoamines (norepinephrine, epinephrine, dopamine, histamine, and serotonin); 3. Peptides (opioid peptides, substance P, somatostatin); and 4. Others (acetylcholine, NO, nucleosides).
Targets for Neuroscience
- 5-HT Receptor(510)
- AChR(57)
- AChE(103)
- Alzheimer(88)
- Amyloid β(130)
- BACE(5)
- CGRP (29)
- COX(286)
- DAPK(5)
- Dopamine Receptor(295)
- GABA Receptor(225)
- Gap Junction(15)
- GluR(121)
- Histamine(2)
- Histamine Receptor(229)
- mPEGS-1(4)
- Muscarinic Receptor(42)
- Neuroscience Peptides(47)
- Nicotinic Receptor(65)
- P2 Receptor(2)
- P2X7 receptor(3)
- SSRIs(7)
- Substance P/NK1 Receptor(20)
- NMDA(2)
- Cholecystokinin Receptor(22)
- GPR139(3)
- mAChR(132)
- MCHR1 (GPR24)(15)
- Neurokinin Receptor(58)
- iGluR(130)
- nAChR(60)
- Beta-secretase(24)
- CaMK(28)
- Dopamine Transporter(17)
- Monoamine Oxidase(78)
- Serotonin Transporter(54)
- Behavioral Neuroscience(274)
- DREADD(0)
- Huntington(10)
- Neuroendocrinology(39)
- Neuroprotection(81)
- Ophthalmology(116)
- Pain Research(166)
- Parkinson(49)
- Seizure Disorders(74)
- Prion(6)
- Cholinesterases(13)
Products for Neuroscience
- Cat.No. 상품명 정보
- GC14752 2,4-Dihydroxyphenylacetyl-L-asparagine glutamate receptors blocker
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GC49159
2-(1-Piperazinyl)pyrimidine
PmP, 1-PP, 1-(2-Pyrimidyl)piperazine
An α2-AR antagonist and active metabolite of azapirones - GC46505 2-(Isopentylamino)naphthalene-1,4-dione A vitamin K analog
- GC17308 2-3-Pyridinedicarboxylic acid
-
GC49481
2-Aminotetralin
2-AT, Tetralin-2-amine
A neuromodulatory agent - GC14873 2-CMDO Dopamine D2-like receptor antagonist
-
GC40473
2-hydroxy Lignoceric Acid
Cerebronic Acid
2-hydroxy Lignoceric acid is an α-hydroxy very long chain fatty acid that is normally present in the mammalian nervous system. - GC11267 2-Hydroxysaclofen 2-하이드록시사클로펜은 강력한 γ-아미노-부티르산-B(GABAB) 수용체 길항제입니다.
- GC38108 2-Methyl-5-HT 2-Methyl-5-HT(2-Methyl-5-hydroxytryptamine)는 강력하고 선택적인 5-HT3 수용체 작용제입니다.
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GC11176
2-Methyl-5-hydroxytryptamine hydrochloride
2-Methyl-5-hydroxytryptamine hydrochloride; 2-Methylserotonin hydrochloride; 2-Me-HT hydrochloride
2-메틸-5-하이드록시트립타민 염산염(2-메틸-5-하이드록시트립타민 염산염)은 강력하고 선택적인 5-HT3 수용체 작용제입니다. -
GC49840
2-Methylbutyrylglycine
2-MBG, N-sec-Valerylglycine
A metabolite of isoleucine -
GC52170
2-Nitroamino-2-imidazoline
NSC 25961, NSC 65424, NSC 91792
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GC11001
2-Pyridylethylamine dihydrochloride
Histamine H1 receptor agonist
- GC14959 2-[1-(4-Piperonyl)piperazinyl]benzothiazole 5-HT4 receptor
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GC42087
21-desacetyl Deflazacort
L-6,485
21-desacetyl Deflazacort is the active glucocorticoid derived from the prodrug deflazacort. -
GC41210
22-HDHA
22-hydroxy Docosahexaenoic Acid, 22-OH DHA
22-HDHA is an oxidation product of docosahexaenoic acid. -
GC40571
24(S),25-epoxy Cholesterol
24(S)-24,25-EC
24(S),25-epoxy Cholesterol is an oxysterol and the most abundant oxysterol in mouse ventral midbrain.
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GC41614
24-dehydro Cholesterol
Desmosterol
24-디히드로콜레스테롤은 콜레스테롤과 유사한 분자입니다.
-
GC46243
24-dehydro Cholesterol-d6
Desmosterol-d6
An internal standard for the quantification of 24-dehydro cholesterol - GC33673 24-Hydroxycholesterol 24-하이드록시콜레스테롤은 N-메틸-d-아스파테이트(NMDA) 수용체R의 양성 알로스테릭 조절제이자 전사 인자 LXR의 강력한 활성화제 역할을 하는 천연 스테롤입니다.
- GC31021 2614W94 2614W94는 기질로 세로토닌을 사용하여 5nM의 IC50 및 1.6nM의 Ki를 억제하는 경쟁 메커니즘을 가진 모노아민 산화효소-A의 선택적 가역적 억제제입니다.
-
GC15856
3'-Fluorobenzylspiperone maleate
ligand for the D2 receptor
- GC15606 3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride dopamine uptake and transport inhibitor
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GC41480
3'-hydroxy Lidocaine
m-hydroxy Lidocaine, meta-hydroxy Lidocaine
3'-hydroxy Lidocaine is an active metabolite of lidocaine formed by the cytochrome P450 (CYP) isoforms CYP1A2 and CYP3A4. -
GC42242
3'-sulfo Galactosylsphingosine (ammonium salt)
Lyso 3’-sulfo Galactosylceramide, Lyso-Sulfatide, Sphingosine-1-Galactoside-3-Sulfate, Sulfogalactosylsphingosine
3'-sulfo Galactosylsphingosine is a form of sulfatide that is lacking the fatty acyl group. -
GC42201
3,3'-Diiodo-L-thyronine
L-3,3'-Diiodothyronine, T2, 3,3'-T2
3,3'-Diiodo-L-thyronine(3,3'-T2)은 갑상선 호르몬의 내인성 대사 산물입니다. - GC33703 3,4,5-Trimethoxycinnamic acid 3,4,5-Trimethoxycinnamic acid는 Polygala tenuifoliaWILLD의 뿌리에서 분리된 페닐프로파노이드로 항스트레스 효과가 있어 동물의 수면 시간을 연장시킵니다.
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GC14343
3,4-dihydro Naratriptan
Naratriptan Impurity B
selective serotonin 5-HT1B agonist - GC46557 3,4-Dihydroquinolin-2(1H)-one A building block
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GC49169
3,8’-Biapigenin
I3,II8-Biapigenin, 3,8\-Biapigenin
3,8’-Biapigenin은 Hypericum perforatum L.의 비플라본입니다. -
GC52324
3-(3-Hydroxyphenyl)propionic Acid sulfate
3-HPPA sulfate
A metabolite of certain phenols and glycosides -
GC42198
3-(4-Chlorophenyl)-4-hydroxybutyric Acid (sodium salt)
γ-Hydroxybaclofen
An inactive metabolite of baclofen -
GC46583
3-Amino-2,6-Piperidinedione
α-Aminoglutarimide, 3-Aminoglutarimide, Glutamimide
An active metabolite of (±)-thalidomide -
GC52129
3-Amino-5-hydroxybenzoic Acid
AHBA
-
GC42248
3-Aminopropylphosphonic Acid
β-Aminopropylphosphonic Acid, 3-APPA, NSC 133832
3-Aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding assay). - GC15569 3-AQC 5-HT3 antagonist
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GC11757
3-Bromocytisine
3-Br-cytisine
3-브로모시티신(3-Br-시티신)은 강력한 nACh 수용체 작용제이며 IC50은 hα4β4, hα4β2 및 hα7-nACh에 대해 각각 0.28, 0.30 및 31.6 nM입니다. - GC12641 3-CPMT dopamine uptake inhibitor
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GC42258
3-Cysteinylacetaminophen (trifluoroacetate salt)
3-(cysteine-S-yl)acetaminophen, APAP-Cys
An acetaminophen-protein adduct - GC60499 3-Hydroxy agomelatine 3-하이드록시 아고멜라틴은 아고멜라틴의 대사 산물입니다.
- GC68328 3-Hydroxy agomelatine-d3
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GC42274
3-hydroxy Darifenacin
UK 148993
3-hydroxy Darifenacin is a metabolite of darifenacin. -
GC41565
3-hydroxy Medetomidine
3-OH Medetomidine, Medetomidine metabolite MIII
3-hydroxy Medetomidine is a metabolite of the α2-adrenergic receptor agonist medetomidine. -
GC18311
3-hydroxy Octanoic Acid
3-hydroxy Caprylic Acid, β-hydroxy Octanoic Acid
3-hydroxy Octanoic acid is a hydroxylated fatty acid that has been found in LPS from P. -
GC40487
3-hydroxy Undecanoic Acid
β-hydroxy Undecanoic Acid
3-hydroxy Undecanoic acid is a hydroxylated fatty acid that has been found in S. -
GC52048
3-hydroxy-4-Methoxyphenethylamine (hydrochloride)
4-O-methyl Dopamine, p-methoxy Dopamine, para-methoxy Dopamine, 4-methoxy-3-Hydroxyphenethylamine
3-히드록시-4-메톡시페네틸아민(염산염)은 디히드로프테리딘 환원효소 억제 효과가 있는 카테콜아민 화합물입니다. -
GC45336
3-hydroxy-DL-Kynurenine
DL-3-Hydroxykynurenine
트립토판의 대사산물인 3-하이드록시-DL-키누레닌은 잠재적인 내인성 신경독이며, 그 수치가 여러 신경퇴행성 장애에서 설명된 바 있습니다. -
GC42294
3-Iodothyronamine (hydrochloride)
T1AM
3-Iodothyronamine is derived from the deiodination and decarboxylation of endogenous thyroxine. - GC11223 3-MATIDA mGlu1 receptor antagonist
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GC49869
3-Methoxytyrosine
DL-3-O-Methyldopa, NSC 122476, 3-methoxy-DL-Tyrosine
An active metabolite of L-DOPA - GC12506 3-Methyl-GABA 3-Methyl-GABA는 강력한 GABA 아미노전이효소 활성화제입니다.
-
GC49149
3-Methylglutaconic Acid
β-Methylglutaconic Acid, 3-MGA, 3-MGC Acid, NSC 249232
A branched-chain organic acid -
GC42307
3-O-methyl-L-DOPA (hydrate)
3-O-methyl-3,4-Dihydroxyphenylalanine, 3-methoxy DOPA, 3-OMD
3-O-methyl-L-DOPA is a metabolite of L-DOPA, produced by the activity of catechol O-methyltransferase. - GC60505 3-O-Methyldopa 3-O-메틸도파(3-메톡시-L-티로신)는 카테콜-O-메틸트랜스퍼라제(COMT)에 의해 형성되는 L-DOPA의 대사 산물입니다.
- GC60506 3-O-Methyldopa D3 3-O-Methyldopa D3(3-Methoxy-L-tyrosine-d3)는 3-O-Methyldopa로 표시된 중수소입니다.
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GC10484
3-pyr-Cytisine
α4β2 receptors agonist
- GC52391 306-O12B-3 An ionizable cationic lipidoid
-
GC18817
3β-hydroxy-5-Cholestenoic Acid
3β-hydroxy-5-CA, Cholesterol-26-carboxylic Acid
3β-hydroxy-5-Cholestenoic acid is an active metabolite of cholesterol formed when cholesterol is metabolized by the cytochrome P450 (CYP) isomer CYP27A1. - GC49367 4’-hydroxy Atomoxetine Glucuronide (hydrate) A metabolite of atomoxetine
- GC49252 4’-hydroxy Trazodone A metabolite of trazodone
- GC40768 4(Z),7(Z),10(Z),13(Z),16(Z)-Nonadecapentaenoic Acid 4(Z),7(Z),10(Z),13(Z),16(Z)-Nonadecapentaenoic acid is an unusual polyunsaturated fatty acid (PUFA) generated during the synthesis of docosahexaenoic acid-d5.
- GC45340 4(Z),7(Z),10(Z),13(Z)-Hexadecatetraenoic Acid
- GC62799 4,4-Diphenylbutylamine hydrochloride 4,4-Diphenylbutylamine은 각각 2589 및 1670 nM의 Kis로 5-HT2A 및 H1 수용체에 대한 친화성을 나타냅니다.
-
GC49752
4,5-Desisopropylidene Topiramate
4,5-Desisopropylidene TPM
An inactive metabolite of topiramate - GC30952 4-(6-Bromo-2-benzothiazolyl)-N-methylbenzenamine 4-(6-브로모-2-벤조티아졸릴)-N-메틸벤젠아민은 1.7 nM의 KD로 아밀로이드-β(1-40)에 결합하는 강력한 아밀로이드 영상화제입니다.
- GC31208 4-(6-Bromo-2-benzothiazolyl)benzenamine 4-(6-Bromo-2-benzothiazolyl)benzenamine은 β-아밀로이드 PET(양전자방출단층촬영) 추적자로서 알츠하이머, 다운증후군과 같은 신경계 질환의 진단에 사용할 수 있습니다.
- GC40045 4-(Dimethylamino)-1-methylpyridinium (iodide) 4-(Dimethylamino)-1-methylpyridinium is a monoquaternary pyridinium salt with anticholinesterase and antiproliferative activities.
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GC33504
4-Acetamidobutanoic acid (N-acetyl GABA)
4-Acetamidobutanoic Acid, N-acetyl-4-Aminobutanoic Acid, N-acetyl-γ-Aminobutyric Acid, NSC 27423
GABA의 주요 대사산물인 4-아세트아미도부탄산(N-아세틸 GABA)(N-아세틸 GABA)은 항산화 및 항균 활성을 나타냅니다. - GC15383 4-Acetyl-1,1-dimethylpiperazinium iodide nicotinic agonist
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GC42338
4-Aminobenzoic Acid hydrazide
4ABAH, Myeloperoxidase Inhibitor 1, NSC 640
4-Aminobenzoic Acid hydrazide는 IC50이 0.3 μ인 비가역적 MPO myeloperoxidase 억제제입니다. - GC49657 4-chloro Trazodone isomer (hydrochloride) An isomer of trazodone
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GC13348
4-DAMP
4-Diphenylacetoxy-N-methyl-piperidine methiodide
4-DAMP는 M3 수용체의 강력한 길항제이며 밀접하게 관련된 M5 수용체에 대해서도 높은 친화력을 가지고 있습니다. -
GC42373
4-epi Minocycline
4-EMC, Minocycline Impurity A
4-epi Minocycline is the main degradation product of and a potential impurity in commercial preparations of minocycline. -
GC48824
4-hydroxy Estrone
4-hydroxy E1, 4-OHE1
에스트론 대사산물인 4-하이드록시 에스트론(4-OHE1)은 산화성 신경독성에 대한 강력한 신경보호 효과가 있습니다. -
GC42411
4-hydroxy Nonenal Alkyne
Click Tag 4HNE Alkyne
4-hydroxy Nonenal (4-HNE) is a major aldehyde produced during the lipid peroxidation of ω-6 polyunsaturated fatty acids, such as arachidonic acid and linoleic acid.
- GC40879 4-hydroxy Solifenacin N-oxide 4-hydroxy Solifenacin N-oxide is an N-oxide form of 4-hydroxy solifenacin, the major metabolite of solifenacin .
-
GC42417
4-hydroxy-3-Methoxyphenylglycol (piperazine salt)
MHPG piperazine, MOPEG piperazine
4-hydroxy-3-Methoxyphenylglycol (piperazine salt) is a metabolite of norepinephrine derived in part by deamination of normetanephrine or by O-methylation of dihydroxyphenylglycol after cellular uptake of either intermediate. - GC60519 4-Hydroxyderricin Angelica keiskei Koidzumi의 주요 활성 성분인 4-Hydroxyderricin은 IC50이 3.43μM인 강력한 선택적 MAO-B(모노아민 산화효소 억제제) 억제제입니다.
- GC63628 4-Hydroxymidazolam
- GC39307 4-Methylamino antipyrine 4-Methylamino 안티피린은 Metamizole의 활성 대사 산물입니다.
-
GC60523
4-Methylamino antipyrine hydrochloride
Metamizole Impurity C
4-Methylamino antipyrine hydrochloride는 Metamizole의 활성 대사 산물입니다. -
GC11606
4-Methylbenzylidene camphor
Enzacamene|Eusolex 6300|4-MBC|Neo Heliopan MBC|Parsol 500|Uvinul MBC 95
4-메틸벤질리덴 장뇌(4-MBC; Enzacamene)는 UV, 특히 UV B 방사선으로부터 피부를 보호하는 능력 때문에 화장품 산업에서 사용되는 유기 장뇌 유도체입니다. - GC12737 4-Methylhistamine dihydrochloride 4-메틸히스타민(2염산염)은 히스타민 4 수용체(H4R)의 강력한 작용제입니다. 4-메틸히스타민(2염산염)은 암 및 자가면역 질환과 같은 면역 관련 질병의 연구에 대한 잠재력이 있습니다.
-
GC42443
4-Methylumbelliferyl 6-thio-Palmitate-β-D-Glucopyranoside
Mu-6S-Palm-β-Glc
4-Methylumbelliferyl 6-thio-Palmitate-β-D-Glucopyranoside는 팔미토일-단백질 티오에스테라제(PPT)에 대한 형광 기질입니다. -
GC40510
4-Methylumbelliferyl-α-D-Galactopyranoside
MU-α-Gal, 4-MU-α-Gal
4-메틸움벨리페릴-α-D-갈락토피라노시드(4MU-α-Gal), α-갈락토시다제 A(GLA)에 대한 기질, 청색 프로-플루오로제닉 기질 -
GC42447
4-Methylumbelliferyl-2-acetamido-2-deoxy-β-D-Glucopyranoside
4-Methylumbelliferyl-N-acetyl-β-Glucosaminide, 4-ΜU-2-acetamido-2-deoxy-β-D-Glucopyranoside
4-Methylumbelliferyl-2-acetamido-2-deoxy-β-D-Glucopyranoside는 N-acetyl-β-D-glucosaminidase에 대한 형광 기질입니다. -
GC49244
4-oxo Isotretinoin
Ro 22-6595
An active metabolite of isotretinoin - GC14311 4-Phenyl-1,2,3,4-tetrahydroisoquinoline hydrochloride dopamine release inhibitor
- GC46675 4-Phenyl-2-pyrrolidinone A precursor and synthetic intermediate
- GC16040 4F 4PP oxalate 4F 4PP(옥살산염)는 선택적 5-HT2A 길항제로서 케탄세린과 거의 같은 높은 친화도(Ki= 5.3 nM)를 갖지만 5-HT2C 부위에 대한 친화도는 훨씬 낮습니다(Ki= 620 nM)[3 ].
-
GC40053
5α,6α-epoxy Cholestanol
NSC 18176
An oxysterol and a metabolite of cholesterol produced by oxidation -
GC46715
5α,6β-Dihydroxycholestanol-d7
Cholestanetriol-d7, 5α,6β-di-OHC-d7
An internal standard for the quantification of 5α,6β-dihydroxycholestanol -
GC48843
5α-Androst-16-en-3α-ol
Androstenol, E 281, NSC 71076
A pheromone with diverse biological activities -
GC49540
5α-Androst-2-ene-17-one
NSC 44506, NSC 80614
A steroid and synthetic intermediate - GC18582 5'-hydroxy Meloxicam A metabolite of meloxicam
- GC60527 5,7-Dimethoxyluteolin 5,7-디메틸루테올린 유도체인 5,7-디메톡시루테올린은 3.417μM의 EC50을 갖는 도파민 수송체(DAT) 활성화제입니다.
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GC14814
5-Carboxamidotryptamine maleate
5-CT maleate
5-HT1 agonist - GC31234 5-HT1A modulator 1 5-HT1A 조절제 1은 각각 2 ±0.3 nM, 10 ± 3 nM 및 40 ±9 nM의 IC50으로 5HT1A, 아드레날린성 α1 및 도파민 D2 수용체에 대해 매우 높은 친화성을 나타냅니다.
- GC60028 5-HT1A modulator 2 hydrochloride 8-OH-DPAT의 유도체인 5-HT1A 조절제 2 염산염은 5-HT1A 결합에 대한 Ki가 53nM인 5-HT1A의 조절제입니다.
- GC32655 5-HT2 antagonist 1 5-HT2 길항제 1은 5-HT2 수용체의 강력한 길항제로, 약한 α1 아드레날린 수용체 차단 활성을 갖는다.