Pain Research
Products for Pain Research
- Cat.No. Product Name Information
- GC49525 Lidocaine-d10 An internal standard for the quantification of lidocaine
- GC47568 Linoleoyl Ethanolamide-d4 An internal standard for the quantification of linoleoyl ethanolamide
- GC48639 Lornoxicam-d4 An internal standard for the quantification of lornoxicam
- GC41181 LY2183240 2'-isomer LY2183240 is a potent, competitive small molecule inhibitor of anandamide uptake (IC50 = 270 pM; Ki = 540 pM) and hydrolysis.
- GC48814 Mesembrine An alkaloid with 5-HT reuptake inhibitory activity
- GC49909 Met-Enkephalinamide (trifluoroacetate salt) A peptide opioid receptor agonist
- GC48907 Metaxalone-d6 An internal standard for the quantification of metaxalone
- GC52049 Myricetin 3-galactoside Myricetin 3-galactoside inhibits xanthine oxidase (XO) activity, lipid peroxidation and scavenges the free radical.
- GC44264 N-(2,6-Dimethylphenyl)-2-(ethylmethylamino)acetamide (hydrochloride) Lidocaine is an anesthetic that blocks voltage-gated Na+ channels (IC50 = 128 μM) with selectivity over L-type Ca2+ channels and GABAA receptors.
- GC18506 N-Arachidonoyl Dopamine N-Arachidonoyl Dopamine is a potent and selective endogenous CB1 receptor agonist with a Ki of 250 nM.
- GC47748 N-Arachidonoyl Dopamine-d8 An internal standard for the quantification of Narachidonoyl dopamine
- GC44319 N-Arachidonoyl-L-Alanine Several different arachidonoyl amino acids, including N-arachidonoyl-L-alanine (NALA), have been isolated and characterized from bovine brain.
- GC41270 N-desmethyl Zolmitriptan N-desmethyl Zolmitriptan (DZT) is an active metabolite of the serotonin (5-HT) receptor subtype 5-HT1B and 5-HT1D agonist zolmitriptan.
- GC47789 N-Oleoyl Glutamine An endogenous N-acyl amine
- GC44442 N-Oleoyl Proline N-Oleoyl proline is an N-acyl amine that has been detected in bovine brain extracts and D.
- GC44456 N-Palmitoyl Glycine N-Palmitoyl Glycine (N-palmitoyl glycine), an endogenous lipid that acts as a modulator of calcium influx and nitric oxide (NO) production in sensory neurons.
- GC47734 Nabumetone-d3 An internal standard for the quantification of nabumetone
- GC49264 Neuromedin U-23 (rat) (trifluoroacetate salt) A peptide NMUR agonist
- GC47768 Neuromedin U-25 (human) (trifluoroacetate salt) A neuropeptide with diverse roles
- GC44387 Neurotensin (trifluoroacetate salt) Neurotensin is a neuropeptide that is distributed throughout the CNS and in enteroendocrine cells of the small intestine that has diverse biological activities.
- GC47788 Nociceptin (trifluoroacetate salt) A neuropeptide
- GC52507 Orexin A amide (bovine, human, mouse, rat) (trifluoroacetate salt) A hypothalamic neuropeptide
- GC49054 Oxaprozin-d5 An internal standard for the quantification of oxaprozin
- GC52342 P4pal10 (trifluoroacetate salt) A PAR4 and FPR2 antagonist and an FFAR2 agonist
- GC44553 Pamoic Acid Pamoic acid is a potent agonist of GPR35 orphan receptors (EC50 = 79 nM in a β-arrestin recruitment assay).
- GC47923 Paraxanthine-d6 An internal standard for the quantification of paraxanthine
- GC49705 Pentapeptide-18 (acetate) A peptide derivative of enkephalin
- GC52177 Perphenazine Sulfoxide
- GC48561 Perphenazine-d4 An internal standard for the quantification of perphenazine
- GC45999 Phentolamine-d4 (hydrochloride) An internal standard for the quantification of phentolamine
- GC49265 PKI (14-22) amide (myristoylated) (trifluoroacetate salt) A PKA inhibitor
- GC49171 Pregabalin Diacid Impurity A potential impurity found in commercial preparations of pregabalin
- GC40184 Probenecid-d14 Probenecid-d14 is intended for use as an internal standard for the quantification of probenecid by GC- or LC-MS.
- GC44687 Prochlorperazine (maleate) Prochlorperazine is a dopamine D2 receptor antagonist with Ki values of 4.7 and 2.9 nM for rat recombinant D2 receptors in CHO cells and rat striatal membranes, respectively.
- GC49120 Prosaptide TX14(A) (trifluoroacetate salt) A peptide fragment of prosaposin and GPR37L1 and GPR37 agonist
- GC48356 Psychotridine An alkaloid with diverse biological activities
- GC18397 R-(-)-α-Methylhistamine (hydrochloride) R-(-)-α-Methylhistamine (hydrochloride) is a potent, selective and brain-penetrant agonist of H3 histamine receptor, with a Kd of 50.3 nM.
- GC44810 Reduced Haloperidol Reduced haloperidol is an active metabolite of haloperidol.
- GC49413 Rizatriptan N-oxide A potential impurity found in commercial preparations of rizatriptan
- GC48583 Rizatriptan-d6 (benzoate salt) An internal standard for the quantification of rizatriptan
- GC45823 Rofecoxib-d5 An internal standard for the quantification of rofecoxib
- GC44857 RWJ 52353 (hydrochloride) An α2D-adrenergic receptor agonist
- GC18650 S-(5'-Adenosyl)-L-methionine (tosylate) S-(5'-Adenosyl)-L-methionine (SAM) is a ubiquitous methyl donor involved in a wide variety of biological reactions, including those mediated by DNA and protein methyltransferases.
- GC44869 Salvinorin A Carbamate Salvinorin A carbamate is a potent κ-opioid receptor (KOR) full agonist that is almost as potent as salvinorin A with EC50 values of 6.2 and 4.5 nM, respectively, for activation of the human KOR to enhance binding of [35S]GTPγS.
- GC44870 Salvinorin A Propionate Salvinorin A propionate is a selective partial agonist at κ1-opioid receptors (KOR) with a Ki value of 32.6 nM.
- GC44871 Salvinorin B Mesylate Salvinorin B mesylate (Mesyl Sal B) is a selective κ-opioid receptor agonist that is more potent than salvinorin A in CHO cells transfected with the human κ-opioid receptor (EC50s = 30 and 40 nM, respectively).
- GC45565 Semax
- GC46221 Seselin An angular pyranocoumarin with diverse biological activities
- GC49112 Sinapyl Alcohol A monolignol with anti-inflammatory and antinociceptive activities
- GC52390 Spexin 1 (human, mouse, rat, bovine) (acetate) An endogenous peptide and agonist of GAL2 and GAL3
- GC48117 Sumatriptan-d6 (succinate) An internal standard for the quantification of sumatriptan
- GC48358 Thymulin (acetate hydrate) A peptide hormone
- GC48178 Tiagabine-d6 (hydrochloride) An internal standard for the quantification of tiagabine
- GC48183 Tizanidine-d4 (hydrochloride) An internal standard for the quantification of tizanidine
- GC48185 Tolperisone-d10 (hydrochloride) An internal standard for the quantification of tolperisone
- GC52005 Triazolomethylindole-3-acetic Acid A metabolite of rizatriptan
- GC52412 TT-232 (trifluoroacetate salt) A synthetic peptide derivative of somatostatin
- GC41599 URB754 URB754 is a potent and noncompetitive inhibitor of monoacylglycerol lipase (MAGL), exhibiting an IC50 value of 200 nM for the recombinant rat brain enzyme.
- GC18923 URB937 A potent FAAH inhibitor
- GC18231 Urocortin II (human) (trifluoroacetate salt) Urocortin II is a neuropeptide hormone and member of the corticotropin-releasing factor (CRF) family which includes mammalian CRF , urocortin , urocortin III , frog sauvagine, and piscine urotensin I.
- GC45139 Vapreotide (trifluoroacetate salt) Vapreotide is a peptide neurokinin-1 receptor (NK1) antagonist and analog of somatostatin (IC50 = 330 nM in a radioligand binding assay).
- GC50671 VCP 171 A positive allosteric modulator of adenosine A1 receptors
- GC45159 WOBE437 WOBE437 is a potent endocannabinoid uptake inhibitor with IC50 values of 10 and 283 nM for arachidonoyl ethanolamide and 2-arachidonoyl glycerol uptake, respectively, in U937 cells.