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GABA Receptor

GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.

Products for  GABA Receptor

  1. Cat.No. Product Name Information
  2. GC38010 γ-Aminobutyric acid γ-Aminobutyric acid  Chemical Structure
  3. GC64508 γ-Aminobutyric acid-d6

    γ-Aminobutyric acid-d6 (4-Aminobutyric acid-d6) is the deuterium labeled γ-Aminobutyric acid.

    γ-Aminobutyric acid-d6  Chemical Structure
  4. GC11449 β-CCB

    benzodiazepine receptor ligand

    β-CCB  Chemical Structure
  5. GC14834 (±)-Nipecotic acid GABA uptake inhibitor (±)-Nipecotic acid  Chemical Structure
  6. GC34954 (+)-Borneol (+)-Borneol  Chemical Structure
  7. GC30933 (+)-Kavain

    An Analytical Reference Standard

    (+)-Kavain  Chemical Structure
  8. GC38677 (-)-α-Pinene (-)-α-Pinene is a monoterpene and shows sleep enhancing property through a direct binding to GABAA-benzodiazepine (BZD) receptors by acting as a partial modulator at the BZD binding site. (-)-α-Pinene  Chemical Structure
  9. GC10065 (-)-Bicuculline methiodide GABAA receptor antagonist (-)-Bicuculline methiodide  Chemical Structure
  10. GC16857 (-)-Bicuculline methobromide (-)-Bicuculline methobromide  Chemical Structure
  11. GC15636 (-)-Bicuculline methochloride (-)-Bicuculline methochloride  Chemical Structure
  12. GC30889 (-)-Securinine An alkaloid (-)-Securinine  Chemical Structure
  13. GC66255 (E)-3,4,5-Trimethoxycinnamic acid (E)-3,4,5-Trimethoxycinnamic acid (TMCA) is a cinnamic acid substituted by multi-methoxy groups. (E)-3,4,5-Trimethoxycinnamic acid is an orally active and potent GABAA/BZ receptor agonist. (E)-3,4,5-Trimethoxycinnamic exhibits favourable binding affinity to 5-HT2C and 5-HT1A receptor, with IC50 values of 2.5 and 7.6 μM, respectively. (E)-3,4,5-Trimethoxycinnamic acid shows anticonvulsant and sedative activity. (E)-3,4,5-Trimethoxycinnamic acid can be used for the research of insomnia, headache and epilepsy. (E)-3,4,5-Trimethoxycinnamic acid  Chemical Structure
  14. GC14111 (R)-baclofen GABA receptor agonist (R)-baclofen  Chemical Structure
  15. GC34986 (R)-Baclofen hydrochloride (R)-Baclofen hydrochloride (Arbaclofen hydrochloride) is a selective GABAB receptor agonist. (R)-Baclofen hydrochloride  Chemical Structure
  16. GC15464 (S)-SNAP 5114 GABA uptake inhibitor (S)-SNAP 5114  Chemical Structure
  17. GC12927 (±)-Baclofen A GABAB agonist (±)-Baclofen  Chemical Structure
  18. GC17223 17-PA GABAA receptor antagonist 17-PA  Chemical Structure
  19. GC11267 2-Hydroxysaclofen GABAB receptor antagonist 2-Hydroxysaclofen  Chemical Structure
  20. GC33703 3,4,5-Trimethoxycinnamic acid 3,4,5-Trimethoxycinnamic acid is a phenylpropanoid isolated from the roots of Polygala tenuifoliaWILLD, with anti-stress effect, prolonging the sleeping time in animals. 3,4,5-Trimethoxycinnamic acid  Chemical Structure
  21. GC12506 3-Methyl-GABA GABA aminotransferase activator 3-Methyl-GABA  Chemical Structure
  22. GC33504 4-Acetamidobutanoic acid (N-acetyl GABA) 4-Acetamidobutanoic acid (N-acetyl GABA) (N-acetyl GABA), the main metabolite of GABA, exhibits antioxidant and antibacterial activities. 4-Acetamidobutanoic acid (N-acetyl GABA)  Chemical Structure
  23. GC30943 6,2'-Dihydroxyflavone 6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor. 6,2'-Dihydroxyflavone  Chemical Structure
  24. GC11284 6-(4-Methoxyphenyl)-3-pyridazinamine GABAA receptor antagonist 6-(4-Methoxyphenyl)-3-pyridazinamine  Chemical Structure
  25. GC30898 6-Methylflavone 6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors. 6-Methylflavone  Chemical Structure
  26. GC10641 AA 29504 GABAA receptor modulator AA 29504  Chemical Structure
  27. GC30844 Afloqualone An Analytical Reference Standard Afloqualone  Chemical Structure
  28. GC14192 Allopregnanolone Allopregnanolone, a 3alpha, 5alpha progesterone metabolite, acts as a potent allosteric modulator of the γ-aminobutyric acid type A (GABAA) receptor, exerts antidepressant and neuroprotective action. Allopregnanolone  Chemical Structure
  29. GC30983 alpha-Asarone (α-Asarone) alpha-Asarone (α-Asarone) (α-Asarone) is one of the main psychoactive compounds, and possesses an antidepressant-like activity in mice. alpha-Asarone (α-Asarone)  Chemical Structure
  30. GC13515 Alphaxalone activates and potentiates GABAA receptor-activated membrane current (IGABA) Alphaxalone  Chemical Structure
  31. GC34064 Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) Aminooxyacetic acid (Carboxymethoxylamine) hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T. Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride)  Chemical Structure
  32. GC63879 Arecaidine hydrochloride Arecaidine hydrochloride, a pyridine alkaloid, is a potent GABA uptake inhibitor. Arecaidine hydrochloride  Chemical Structure
  33. GC10974 AWD 131-138 AWD 131-138 (AWD 131-138) is a new low-affinity partial benzodiazepine receptor agonist with potent anticonvulsant and anxiolytic properties in rodent models. AWD 131-138  Chemical Structure
  34. GC31010 AZD-6280 AZD-6280 is a selective GABAA(α2/3) receptor modulator, used for treatment of generalized anxiety disorder. AZD-6280  Chemical Structure
  35. GC31990 Bamaluzole Bamaluzole is a GABA receptor agonist extracted from patent WO 2012064642 A1. Bamaluzole  Chemical Structure
  36. GC19057 Basmisanil Basmisanil is a highly selective GABAAα5 negative allosteric modulator. Basmisanil  Chemical Structure
  37. GC12414 Bemegride GABA receptor antagonist Bemegride  Chemical Structure
  38. GC34494 Bifenazate An acaricide Bifenazate  Chemical Structure
  39. GC11565 Bretazenil GABAA benzodiazepine site partial agonist Bretazenil  Chemical Structure
  40. GC30521 Broflanilide Broflanilide is a potential insecticide and metabolized to Desmethyl-Broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin (RDL) GABA Receptor, and inhibits S. Broflanilide  Chemical Structure
  41. GC31224 Carburazepam (RGH 3331) Carburazepam (RGH 3331) is a drug which derives from benzodiazepine. Carburazepam (RGH 3331)  Chemical Structure
  42. GC13374 CGP 13501 Positive modulator of GABAB receptors,allosteric CGP 13501  Chemical Structure
  43. GC11153 CGP 35348 Selective GABAB antagonist, brain penetrant CGP 35348  Chemical Structure
  44. GC13676 CGP 36216 hydrochloride Selective GABAB antagonist CGP 36216 hydrochloride  Chemical Structure
  45. GC35669 CGP 36742 CGP 36742 is a selective GABAB receptor antagonist that can penetrate the blood–brain barrier after peripheral administration, with an IC50 of 32?μM. CGP 36742  Chemical Structure
  46. GC13131 CGP 46381 GABAB receptor antagonist CGP 46381  Chemical Structure
  47. GC16947 CGP 52432 GABAB receptor antagonist CGP 52432  Chemical Structure
  48. GC10489 CGP 54626 hydrochloride

    GABAB receptor antagonist

    CGP 54626 hydrochloride  Chemical Structure
  49. GC16600 CGP 55845 hydrochloride GABAB receptor antagonist CGP 55845 hydrochloride  Chemical Structure
  50. GC15563 CGP 7930 Positive allosteric modulator of GABAB receptors CGP 7930  Chemical Structure
  51. GC33751 CGP11952 CGP11952 is a triazolyl-Benzaphenon resembling the benzodiazepines in its pharmacological action. CGP11952  Chemical Structure
  52. GC14274 CGS 20625 partial agonist for the benzodiazepine binding site of the GABAA receptor CGS 20625  Chemical Structure
  53. GC16311 Chlormethiazole hydrochloride GABAA agonist Chlormethiazole hydrochloride  Chemical Structure
  54. GC16691 Chlormezanone Anxiolytic and skeletal muscle relaxant Chlormezanone  Chemical Structure
  55. GC43261 Cholesteryl Myristate Cholesteryl Myristate is a natural steroid present in traditional Chinese medicine. Cholesteryl Myristate binds to several ion channels such as the nicotinic acetylcholine receptor, GABAA receptor, and the inward-rectifier potassium ion channel. Cholesteryl Myristate  Chemical Structure
  56. GC14477 CI 966 hydrochloride GABA transporter GAT-1 inhibitor CI 966 hydrochloride  Chemical Structure
  57. GC31120 Cirsimaritin Cirsimaritin binds weakly to the benzodiazepine site on GABAA receptors, with antidepressant, anxiolytic and antinociceptive activities. Cirsimaritin  Chemical Structure
  58. GC16188 CL 218872 Benzodiazepine agonist CL 218872  Chemical Structure
  59. GC38758 Clomethiazole Chlormethiazole is an potent and orally active GABAA?agonist. Clomethiazole  Chemical Structure
  60. GC31052 CP-409092 CP-409092 is a partial agonist of GABAA receptor, with anti-anxiety activity. CP-409092  Chemical Structure
  61. GC38387 CP-409092 hydrochloride CP-409092 hydrochloride is a partial agonist of GABAA receptor, with anti-anxiety activity. CP-409092 hydrochloride  Chemical Structure
  62. GC30930 DAA-1106 A TSPO agonist DAA-1106  Chemical Structure
  63. GC10530 Dihydroergotoxine mesylate GABAA receptor modulator Dihydroergotoxine mesylate  Chemical Structure
  64. GC13405 DMCM hydrochloride Benzodiazepine inverse agonist DMCM hydrochloride  Chemical Structure
  65. GC14150 DPNI-caged-GABA

    activates GABAA receptor

    DPNI-caged-GABA  Chemical Structure
  66. GC12008 DS2 Positive allosteric modulator of δ-subunit containing GABAA receptors DS2  Chemical Structure
  67. GC35975 Emamectin Benzoate Emamectin Benzoate (MK-244) is an orally active nervoussystem toxicant by binding g-aminobutyric (GABA) receptor in insects. Emamectin Benzoate  Chemical Structure
  68. GC64673 Etbicyphat Etbicyphat (Trimethylopropane phosphate) is a potent GABA(A) receptors competitive antagonist. Etbicyphat  Chemical Structure
  69. GC31023 Ethyl dirazepate Ethyl dirazepate is a drug which is a benzodiazepine derivative. Ethyl dirazepate  Chemical Structure
  70. GC36012 Etifoxine A positive allosteric modulator of GABAA receptors Etifoxine  Chemical Structure
  71. GC16134 Etomidate

    General anesthetic with GABA modulatory and GABA-mimetic actions

    Etomidate  Chemical Structure
  72. GC16985 Etomidate hydrochloride

    GABAA receptors agonist

    Etomidate hydrochloride  Chemical Structure
  73. GC12568 FG 7142 benzodiazepine inverse agonist and anxiogenic agent FG 7142  Chemical Structure
  74. GC33754 FG8119 (NNC13-8119) FG8119 (NNC13-8119) is a novel benzodiazepine agonist extracted from patent US 4745112 A. FG8119 (NNC13-8119)  Chemical Structure
  75. GC14017 FGIN-1-27

    high affinity agonist of the translocator protein (TSPO,peripheral benzodiazepine receptor)

    FGIN-1-27  Chemical Structure
  76. GC16238 FGIN-1-43 ligand as probe for the mitochondial DBI receptor (peripheral benzodiazepine receptor) FGIN-1-43  Chemical Structure
  77. GC10772 Flumazenil

    Benzodiazepine antagonist

    Flumazenil  Chemical Structure
  78. GC36058 Flumazenil acid Flumazenil acid is a metabolite of Flumazenil. Flumazenil acid  Chemical Structure
  79. GC30088 Fluxametamide Fluxametamide is an insecticide with wide spectrum, acts as an antagonist of GABA- and glutamate-gated chloride channels, with IC50 of 1.95 nM and 225 nM for M. Fluxametamide  Chemical Structure
  80. GC12714 Gabapentin

    GABA enhancer

    Gabapentin  Chemical Structure
  81. GC38543 Gaboxadol hydrochloride A GABAA receptor agonist and GABAC receptor antagonist Gaboxadol hydrochloride  Chemical Structure
  82. GC11156 Ganaxolone positive allosteric modulator of GABAA receptor Ganaxolone  Chemical Structure
  83. GC16495 GBLD 345 GABAA receptor agonist GBLD 345  Chemical Structure
  84. GC69161 Gidazepam

    Gidazepam is a GABA receptor channel (GABA RCs) agonist.

    Gidazepam  Chemical Structure
  85. GC31205 Gidazepam (Gidasepam)

    Gidazepam is an agonist of GABA receptor channels (GABA RCs).

    Gidazepam (Gidasepam)  Chemical Structure
  86. GC11303 GS 39783 Positive allosteric modulator of GABAB receptor GS 39783  Chemical Structure
  87. GC14659 Guvacine hydrochloride GABA uptake inhibitor Guvacine hydrochloride  Chemical Structure
  88. GC12359 Hispidulin Partial positive allosteric modulator at the benzodiazepine receptor Hispidulin  Chemical Structure
  89. GC63950 Homocarnosine TFA Homocarnosine TFA is a dipeptide of γ-aminobutyric acid (GABA) and histidine unique to brain. Homocarnosine TFA  Chemical Structure
  90. GC13567 Isoguvacine hydrochloride

    GABAA receptor agonist

    Isoguvacine hydrochloride  Chemical Structure
  91. GC25531 Isonipecotic acid Isonipecotic acid (4-Piperidinecarboxylic acid, 4-Carboxypiperidine, Hexahydroisonicotinic acid) is a heterocyclic compound that mainly acts as a GABAA receptor partial agonist. Isonipecotic acid  Chemical Structure
  92. GC17350 L-655,708 inverse agonist for the benzodiazepine site of GABAA receptors containing the α5 subunit L-655,708  Chemical Structure
  93. GC11597 L-838,417 Subtype-selective GABAA receptor partial agonist L-838,417  Chemical Structure
  94. GC30862 L-Cycloserine ((S)-4-Amino-3-isoxazolidone) L-Cycloserine ((S)-4-Amino-3-isoxazolidone) ((S)-4-Amino-3-isoxazolidone) irreversibly inhibits GABA pyridoxal 5′-phosphate-dependent aminitransferase in E. L-Cycloserine ((S)-4-Amino-3-isoxazolidone)  Chemical Structure
  95. GC25566 L-DAB HBR L-DAB HBR  Chemical Structure
  96. GC44040 LAU159 A positive allosteric modulator of α6β3γ2 subunit-containing GABAA receptors LAU159  Chemical Structure
  97. GC14045 Loreclezole GABAA receptor modulator Loreclezole  Chemical Structure
  98. GC18299 Lorediplon Lorediplon is a ligand for α1 subunit-containing GABAA receptors. Lorediplon  Chemical Structure
  99. GC65292 Lotilaner Lotilaner is a parasiticide, acts as a potent non-competitive antagonist of insects GABACl receptors, with an IC50 of 23.84 nM for Drosophila melanogaster GABA receptor. Lotilaner  Chemical Structure
  100. GC13715 MK 0343 GABAA partial agonist MK 0343  Chemical Structure
  101. GC16528 MRK 016 GABAA receptor inverse agonist MRK 016  Chemical Structure

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