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Home >> Signaling Pathways >> Membrane Transporter/Ion Channel >> GABA Receptor

GABA Receptor

GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.

Products for  GABA Receptor

  1. Cat.No. Product Name Information
  2. GC74347 α-Casozepine α-Casozepine is a bioactive peptide derived from the α protein S1 casein in milk and has an affinity for γ-aminobutyric acid (GABA) receptors in the brain. α-Casozepine Chemical Structure
  3. GC70650 γ-Acetylenic GABA hydrochloride γ-Acetylenic GABA (GAG) hydrochloride is an irreversible inhibitor of GABA-transaminase. γ-Acetylenic GABA hydrochloride Chemical Structure
  4. GC38010 γ-Aminobutyric acid γ-Aminobutyric acid Chemical Structure
  5. GC64508 γ-Aminobutyric acid-d6

    γ-Aminobutyric acid-d6 (4-Aminobutyric acid-d6) is the deuterium labeled γ-Aminobutyric acid.

     γ-Aminobutyric acid-d6 Chemical Structure
  6. GC11449 β-CCB

    benzodiazepine receptor ligand

     β-CCB Chemical Structure
  7. GC14834 (±)-Nipecotic acid

    (±)-Nipecotic Acid, (R,S)-Nipecotic Acid, 3-Piperidine Carboxylic Acid, DL-Piperidine 3-Carboxylic Acid

     GABA uptake inhibitor (±)-Nipecotic acid Chemical Structure
  8. GC34954 (+)-Borneol

    D-Borneol, (1R)-(+)-Borneol, (+)-endo-Borneol

     (+)-Borneol Chemical Structure
  9. GC30933 (+)-Kavain

    Kawain, NSC 112162

    An Analytical Reference Standard

     (+)-Kavain Chemical Structure
  10. GC38677 (-)-α-Pinene

    NSC 7727

     (-)-α-Pinene is a monoterpene and shows sleep enhancing property through a direct binding to GABAA-benzodiazepine (BZD) receptors by acting as a partial modulator at the BZD binding site. (-)-α-Pinene Chemical Structure
  11. GC10065 (-)-Bicuculline methiodide GABAA receptor antagonist (-)-Bicuculline methiodide Chemical Structure
  12. GC16857 (-)-Bicuculline methobromide (-)-Bicuculline methobromide Chemical Structure
  13. GC15636 (-)-Bicuculline methochloride (-)-Bicuculline methochloride Chemical Structure
  14. GC30889 (-)-Securinine

    NSC 107413, L-Securinine

     An alkaloid (-)-Securinine Chemical Structure
  15. GC66255 (E)-3,4,5-Trimethoxycinnamic acid

    TMCA

     (E)-3,4,5-Trimethoxycinnamic acid (TMCA) is a cinnamic acid substituted by multi-methoxy groups. (E)-3,4,5-Trimethoxycinnamic acid is an orally active and potent GABAA/BZ receptor agonist. (E)-3,4,5-Trimethoxycinnamic exhibits favourable binding affinity to 5-HT2C and 5-HT1A receptor, with IC50 values of 2.5 and 7.6 μM, respectively. (E)-3,4,5-Trimethoxycinnamic acid shows anticonvulsant and sedative activity. (E)-3,4,5-Trimethoxycinnamic acid can be used for the research of insomnia, headache and epilepsy. (E)-3,4,5-Trimethoxycinnamic acid Chemical Structure
  16. GC14111 (R)-baclofen GABA receptor agonist (R)-baclofen Chemical Structure
  17. GC34986 (R)-Baclofen hydrochloride

    (R)-Baclofen

     (R)-Baclofen hydrochloride (Arbaclofen hydrochloride) is a selective GABAB receptor agonist. (R)-Baclofen hydrochloride Chemical Structure
  18. GC15464 (S)-SNAP 5114 GABA uptake inhibitor (S)-SNAP 5114 Chemical Structure
  19. GC12927 (±)-Baclofen A GABAB agonist (±)-Baclofen Chemical Structure
  20. GC17223 17-PA GABAA receptor antagonist 17-PA Chemical Structure
  21. GC70652 2'MeO6MF 2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors. 2'MeO6MF Chemical Structure
  22. GC11267 2-Hydroxysaclofen GABAB receptor antagonist 2-Hydroxysaclofen Chemical Structure
  23. GC33703 3,4,5-Trimethoxycinnamic acid 3,4,5-Trimethoxycinnamic acid is a phenylpropanoid isolated from the roots of Polygala tenuifoliaWILLD, with anti-stress effect, prolonging the sleeping time in animals. 3,4,5-Trimethoxycinnamic acid Chemical Structure
  24. GC12506 3-Methyl-GABA GABA aminotransferase activator 3-Methyl-GABA Chemical Structure
  25. GC33504 4-Acetamidobutanoic acid (N-acetyl GABA)

    4-Acetamidobutanoic Acid, N-acetyl-4-Aminobutanoic Acid, N-acetyl-γ-Aminobutyric Acid, NSC 27423

     4-Acetamidobutanoic acid (N-acetyl GABA) (N-acetyl GABA), the main metabolite of GABA, exhibits antioxidant and antibacterial activities. 4-Acetamidobutanoic acid (N-acetyl GABA) Chemical Structure
  26. GC30943 6,2'-Dihydroxyflavone 6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor. 6,2'-Dihydroxyflavone Chemical Structure
  27. GC11284 6-(4-Methoxyphenyl)-3-pyridazinamine GABAA receptor antagonist 6-(4-Methoxyphenyl)-3-pyridazinamine Chemical Structure
  28. GC30898 6-Methylflavone 6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors. 6-Methylflavone Chemical Structure
  29. GC10641 AA 29504 GABAA receptor modulator AA 29504 Chemical Structure
  30. GC30844 Afloqualone

    HQ-495

     An Analytical Reference Standard Afloqualone Chemical Structure
  31. GC14192 Allopregnanolone

    ALLO, 3α,5α-tetrahydro Progesterone, 3α,5α-THP; brexanolone

     Allopregnanolone, a 3alpha, 5alpha progesterone metabolite, acts as a potent allosteric modulator of the γ-aminobutyric acid type A (GABAA) receptor, exerts antidepressant and neuroprotective action. Allopregnanolone Chemical Structure
  32. GC30983 alpha-Asarone (α-Asarone)

    transAsarone

     alpha-Asarone (α-Asarone) (α-Asarone) is one of the main psychoactive compounds, and possesses an antidepressant-like activity in mice. alpha-Asarone (α-Asarone) Chemical Structure
  33. GC13515 Alphaxalone activates and potentiates GABAA receptor-activated membrane current (IGABA) Alphaxalone Chemical Structure
  34. GC34064 Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride)

    Aminooxyacetate

     Aminooxyacetic acid (Carboxymethoxylamine) hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T. Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) Chemical Structure
  35. GC68659 Anisatin

    Anisatin is a toxic substance isolated from the seeds of a Japanese plant (Illicium anisatum). It is a non-competitive b>GABA antagonist and belongs to the class of convulsant toxins. Anisatin inhibits GABA-induced currents in a concentration-dependent manner, with an EC50 of approximately 1.10 μM.

     Anisatin Chemical Structure
  36. GC63879 Arecaidine hydrochloride Arecaidine hydrochloride, a pyridine alkaloid, is a potent GABA uptake inhibitor. Arecaidine hydrochloride Chemical Structure
  37. GC10974 AWD 131-138

    ELB138, Imepitoin

     AWD 131-138 (AWD 131-138) is a new low-affinity partial benzodiazepine receptor agonist with potent anticonvulsant and anxiolytic properties in rodent models. AWD 131-138 Chemical Structure
  38. GC31010 AZD-6280 AZD-6280 is a selective GABAA(α2/3) receptor modulator, used for treatment of generalized anxiety disorder. AZD-6280 Chemical Structure
  39. GC31990 Bamaluzole Bamaluzole is a GABA receptor agonist extracted from patent WO 2012064642 A1. Bamaluzole Chemical Structure
  40. GC19057 Basmisanil

    RG-1662

     Basmisanil is a highly selective GABAAα5 negative allosteric modulator. Basmisanil Chemical Structure
  41. GC12414 Bemegride GABA receptor antagonist Bemegride Chemical Structure
  42. GC34494 Bifenazate An acaricide Bifenazate Chemical Structure
  43. GC68798 BPDBA

    BPDBA is a selective and non-competitive inhibitor of betaine/GABA transporter (BGT-1), with IC50 values of 20 μM for human BGT-1 and 35 μM for mouse GAT2.

     BPDBA Chemical Structure
  44. GC11565 Bretazenil

    Ro 16-6028

     GABAA benzodiazepine site partial agonist Bretazenil Chemical Structure
  45. GC30521 Broflanilide Broflanilide is a potential insecticide and metabolized to Desmethyl-Broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin (RDL) GABA Receptor, and inhibits S. Broflanilide Chemical Structure
  46. GC31224 Carburazepam (RGH 3331) Carburazepam (RGH 3331) is a drug which derives from benzodiazepine. Carburazepam (RGH 3331) Chemical Structure
  47. GC13374 CGP 13501 Positive modulator of GABAB receptors,allosteric CGP 13501 Chemical Structure
  48. GC11153 CGP 35348 Selective GABAB antagonist, brain penetrant CGP 35348 Chemical Structure
  49. GC13676 CGP 36216 hydrochloride Selective GABAB antagonist CGP 36216 hydrochloride Chemical Structure
  50. GC35669 CGP 36742

    3-Aminopropyl-n-butylphosphinic Acid, SGS 742

     CGP 36742 is a selective GABAB receptor antagonist that can penetrate the blood–brain barrier after peripheral administration, with an IC50 of 32?μM. CGP 36742 Chemical Structure
  51. GC13131 CGP 46381 GABAB receptor antagonist CGP 46381 Chemical Structure
  52. GC16947 CGP 52432 GABAB receptor antagonist CGP 52432 Chemical Structure
  53. GC10489 CGP 54626 hydrochloride

    CGP 54626A

    GABAB receptor antagonist

     CGP 54626 hydrochloride Chemical Structure
  54. GC16600 CGP 55845 hydrochloride GABAB receptor antagonist CGP 55845 hydrochloride Chemical Structure
  55. GC15563 CGP 7930 Positive allosteric modulator of GABAB receptors CGP 7930 Chemical Structure
  56. GC33751 CGP11952 CGP11952 is a triazolyl-Benzaphenon resembling the benzodiazepines in its pharmacological action. CGP11952 Chemical Structure
  57. GC14274 CGS 20625 partial agonist for the benzodiazepine binding site of the GABAA receptor CGS 20625 Chemical Structure
  58. GC16311 Chlormethiazole hydrochloride

    Clomethiazole

     GABAA agonist Chlormethiazole hydrochloride Chemical Structure
  59. GC16691 Chlormezanone

    (±)-Chlormezanone, NSC 169108

     Anxiolytic and skeletal muscle relaxant Chlormezanone Chemical Structure
  60. GC43261 Cholesteryl Myristate

    Cholesterol Myristate, Cholesteryl Tetradecanoate, Myristic Acid cholesteryl ester, NSC 226867

     Cholesteryl Myristate is a natural steroid present in traditional Chinese medicine. Cholesteryl Myristate binds to several ion channels such as the nicotinic acetylcholine receptor, GABAA receptor, and the inward-rectifier potassium ion channel. Cholesteryl Myristate Chemical Structure
  61. GC14477 CI 966 hydrochloride GABA transporter GAT-1 inhibitor CI 966 hydrochloride Chemical Structure
  62. GC31120 Cirsimaritin

    5,4'-Dihydroxy-6,7-dimethoxyflavone

     Cirsimaritin is a dimethoxy flavonoid found in plants, it has anticancer potential and shows potent antimicrobial, antioxidant, antispasmodic, activity, and also inhibits cyclooxygenase-1. Cirsimaritin Chemical Structure
  63. GC16188 CL 218872 Benzodiazepine agonist CL 218872 Chemical Structure
  64. GC38758 Clomethiazole Chlormethiazole is an potent and orally active GABAA?agonist. Clomethiazole Chemical Structure
  65. GC31052 CP-409092 CP-409092 is a partial agonist of GABAA receptor, with anti-anxiety activity. CP-409092 Chemical Structure
  66. GC38387 CP-409092 hydrochloride CP-409092 hydrochloride is a partial agonist of GABAA receptor, with anti-anxiety activity. CP-409092 hydrochloride Chemical Structure
  67. GC30930 DAA-1106 A TSPO agonist DAA-1106 Chemical Structure
  68. GC10530 Dihydroergotoxine mesylate GABAA receptor modulator Dihydroergotoxine mesylate Chemical Structure
  69. GC13405 DMCM hydrochloride Benzodiazepine inverse agonist DMCM hydrochloride Chemical Structure
  70. GC14150 DPNI-caged-GABA

    activates GABAA receptor

     DPNI-caged-GABA Chemical Structure
  71. GC12008 DS2 Positive allosteric modulator of δ-subunit containing GABAA receptors DS2 Chemical Structure
  72. GC35975 Emamectin Benzoate Emamectin Benzoate (MK-244) is an orally active nervoussystem toxicant by binding g-aminobutyric (GABA) receptor in insects. Emamectin Benzoate Chemical Structure
  73. GC64673 Etbicyphat

    Trimethylopropane phosphate

     Etbicyphat (Trimethylopropane phosphate) is a potent GABA(A) receptors competitive antagonist. Etbicyphat Chemical Structure
  74. GC31023 Ethyl dirazepate Ethyl dirazepate is a drug which is a benzodiazepine derivative. Ethyl dirazepate Chemical Structure
  75. GC36012 Etifoxine

    Etafenoxine, HOE 36801

     A positive allosteric modulator of GABAA receptors Etifoxine Chemical Structure
  76. GC16134 Etomidate

    (+)-Etomidate, d-Etomidate, R 16659

    General anesthetic with GABA modulatory and GABA-mimetic actions

     Etomidate Chemical Structure
  77. GC16985 Etomidate hydrochloride

    GABAA receptors agonist

     Etomidate hydrochloride Chemical Structure
  78. GC70546 Fengabine Fengabine is a GABAergic antidepressant agent. Fengabine Chemical Structure
  79. GC12568 FG 7142

    ZK 39106

     benzodiazepine inverse agonist and anxiogenic agent FG 7142 Chemical Structure
  80. GC33754 FG8119 (NNC13-8119)

    NNC13-8119

     FG8119 (NNC13-8119) is a novel benzodiazepine agonist extracted from patent US 4745112 A. FG8119 (NNC13-8119) Chemical Structure
  81. GC14017 FGIN-1-27

    high affinity agonist of the translocator protein (TSPO,peripheral benzodiazepine receptor)

     FGIN-1-27 Chemical Structure
  82. GC16238 FGIN-1-43 ligand as probe for the mitochondial DBI receptor (peripheral benzodiazepine receptor) FGIN-1-43 Chemical Structure
  83. GC70576 Fipronil sulfone Fipronil sulfone is the major metabolite of Fipronil. Fipronil sulfone Chemical Structure
  84. GC10772 Flumazenil

    Ro 1722, Ro 15-1788, Ro 41-8157

    Benzodiazepine antagonist

     Flumazenil Chemical Structure
  85. GC36058 Flumazenil acid Flumazenil acid is a metabolite of Flumazenil. Flumazenil acid Chemical Structure
  86. GC30088 Fluxametamide Fluxametamide is an insecticide with wide spectrum, acts as an antagonist of GABA- and glutamate-gated chloride channels, with IC50 of 1.95 nM and 225 nM for M. Fluxametamide Chemical Structure
  87. GC12714 Gabapentin

    CI-945

    GABA enhancer

     Gabapentin Chemical Structure
  88. GC38543 Gaboxadol hydrochloride A GABAA receptor agonist and GABAC receptor antagonist Gaboxadol hydrochloride Chemical Structure
  89. GC11156 Ganaxolone

    CCD 1042

     positive allosteric modulator of GABAA receptor Ganaxolone Chemical Structure
  90. GC16495 GBLD 345 GABAA receptor agonist GBLD 345 Chemical Structure
  91. GC69161 Gidazepam

    Gidasepam; Hidazepam; Hydazepam

    Gidazepam is a GABA receptor channel (GABA RCs) agonist.

     Gidazepam Chemical Structure
  92. GC31205 Gidazepam (Gidasepam)

    Gidazepam is an agonist of GABA receptor channels (GABA RCs).

     Gidazepam (Gidasepam) Chemical Structure
  93. GC11303 GS 39783 Positive allosteric modulator of GABAB receptor GS 39783 Chemical Structure
  94. GC14659 Guvacine hydrochloride GABA uptake inhibitor Guvacine hydrochloride Chemical Structure
  95. GC12359 Hispidulin

    Dinatin, 6-Methoxyapigenin, NSC 122415

     Partial positive allosteric modulator at the benzodiazepine receptor Hispidulin Chemical Structure
  96. GC63950 Homocarnosine TFA

    L-Homocarnosine TFA; γ-Aminobutyryl-L-histidine TFA

     Homocarnosine TFA is a dipeptide of γ-aminobutyric acid (GABA) and histidine unique to brain. Homocarnosine TFA Chemical Structure
  97. GC70542 HZ166 HZ166 is a GABAA receptor subtype-selective benzodiazepine site agonist with preferential activity at α2- and α3-GABAA receptors. HZ166 Chemical Structure
  98. GC70613 Inaperisone Inaperisone is a centrally acting muscle relaxant. Inaperisone Chemical Structure
  99. GC13567 Isoguvacine hydrochloride

    GABAA receptor agonist

     Isoguvacine hydrochloride Chemical Structure
  100. GC25531 Isonipecotic acid

    4-Piperidinecarboxylic acid, 4-Carboxypiperidine, Hexahydroisonicotinic acid

     Isonipecotic acid (4-Piperidinecarboxylic acid, 4-Carboxypiperidine, Hexahydroisonicotinic acid) is a heterocyclic compound that mainly acts as a GABAA receptor partial agonist. Isonipecotic acid Chemical Structure
  101. GC74052 KGP-25 KGP-25 is an inhibitor of voltage-gated sodium channel 1.8 (Nav1.8), which can be used for analgesia by targeting Nav1.8 in the peripheral nervous system (PNS). KGP-25 Chemical Structure

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