Search Site
  • 0
    My Cart

    Click Here to Find How Many Items You Have Added:)

    image loader

    Adding item(s) to cart......

Home >> Signaling Pathways >> Neuroscience >> GABA Receptor

GABA Receptor

GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.

Products for  GABA Receptor

  1. Cat.No. Product Name Information
  2. GC63615 α-Thujone α-Thujone is a monoterpene isolated from Thuja occidentalis essential oil with potent anti-tumor activities. α-Thujone Chemical Structure
  3. GC38010 γ-Aminobutyric acid γ-Aminobutyric acid Chemical Structure
  4. GC64508 γ-Aminobutyric acid-d6

    γ-Aminobutyric acid-d6 (4-Aminobutyric acid-d6) is the deuterium labeled γ-Aminobutyric acid.

     γ-Aminobutyric acid-d6 Chemical Structure
  5. GC11449 β-CCB

    benzodiazepine receptor ligand

     β-CCB Chemical Structure
  6. GC14834 (±)-Nipecotic acid GABA uptake inhibitor (±)-Nipecotic acid Chemical Structure
  7. GN10745 (+)-Bicuculline

    (+)-Bicuculline is a light-sensitive competitive antagonist of GABA-A receptor.

     (+)-Bicuculline Chemical Structure
  8. GC34954 (+)-Borneol (+)-Borneol Chemical Structure
  9. GC30933 (+)-Kavain

    An Analytical Reference Standard

     (+)-Kavain Chemical Structure
  10. GC38677 (-)-α-Pinene (-)-α-Pinene is a monoterpene and shows sleep enhancing property through a direct binding to GABAA-benzodiazepine (BZD) receptors by acting as a partial modulator at the BZD binding site. (-)-α-Pinene Chemical Structure
  11. GC10065 (-)-Bicuculline methiodide GABAA receptor antagonist (-)-Bicuculline methiodide Chemical Structure
  12. GC16857 (-)-Bicuculline methobromide (-)-Bicuculline methobromide Chemical Structure
  13. GC15636 (-)-Bicuculline methochloride (-)-Bicuculline methochloride Chemical Structure
  14. GC30889 (-)-Securinine An alkaloid (-)-Securinine Chemical Structure
  15. GC60000 (2S)-6-Prenylnaringenin (2S)-6-Prenylnaringenin is the most efficient compound in forebrain. (2S)-6-Prenylnaringenin Chemical Structure
  16. GC66255 (E)-3,4,5-Trimethoxycinnamic acid (E)-3,4,5-Trimethoxycinnamic acid (TMCA) is a cinnamic acid substituted by multi-methoxy groups. (E)-3,4,5-Trimethoxycinnamic acid is an orally active and potent GABAA/BZ receptor agonist. (E)-3,4,5-Trimethoxycinnamic exhibits favourable binding affinity to 5-HT2C and 5-HT1A receptor, with IC50 values of 2.5 and 7.6 μM, respectively. (E)-3,4,5-Trimethoxycinnamic acid shows anticonvulsant and sedative activity. (E)-3,4,5-Trimethoxycinnamic acid can be used for the research of insomnia, headache and epilepsy. (E)-3,4,5-Trimethoxycinnamic acid Chemical Structure
  17. GC14111 (R)-baclofen GABA receptor agonist (R)-baclofen Chemical Structure
  18. GC34986 (R)-Baclofen hydrochloride (R)-Baclofen hydrochloride (Arbaclofen hydrochloride) is a selective GABAB receptor agonist. (R)-Baclofen hydrochloride Chemical Structure
  19. GC15464 (S)-SNAP 5114 GABA uptake inhibitor (S)-SNAP 5114 Chemical Structure
  20. GC12927 (±)-Baclofen A GABAB agonist (±)-Baclofen Chemical Structure
  21. GC17223 17-PA GABAA receptor antagonist 17-PA Chemical Structure
  22. GC60017 2'-O-Methylisoliquiritigenin 2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-regulates 5-HT, NE, DA and GABA pathways, but does not put a very significant effect on ne NE pathway. 2'-O-Methylisoliquiritigenin Chemical Structure
  23. GC11267 2-Hydroxysaclofen GABAB receptor antagonist 2-Hydroxysaclofen Chemical Structure
  24. GC33703 3,4,5-Trimethoxycinnamic acid 3,4,5-Trimethoxycinnamic acid is a phenylpropanoid isolated from the roots of Polygala tenuifoliaWILLD, with anti-stress effect, prolonging the sleeping time in animals. 3,4,5-Trimethoxycinnamic acid Chemical Structure
  25. GC12506 3-Methyl-GABA GABA aminotransferase activator 3-Methyl-GABA Chemical Structure
  26. GC33504 4-Acetamidobutanoic acid (N-acetyl GABA) 4-Acetamidobutanoic acid (N-acetyl GABA) (N-acetyl GABA), the main metabolite of GABA, exhibits antioxidant and antibacterial activities. 4-Acetamidobutanoic acid (N-acetyl GABA) Chemical Structure
  27. GC63628 4-Hydroxymidazolam 4-Hydroxymidazolam Chemical Structure
  28. GC30943 6,2'-Dihydroxyflavone 6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor. 6,2'-Dihydroxyflavone Chemical Structure
  29. GC11284 6-(4-Methoxyphenyl)-3-pyridazinamine GABAA receptor antagonist 6-(4-Methoxyphenyl)-3-pyridazinamine Chemical Structure
  30. GC30898 6-Methylflavone 6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors. 6-Methylflavone Chemical Structure
  31. GC10641 AA 29504 GABAA receptor modulator AA 29504 Chemical Structure
  32. GC14916 Acamprosate calcium An NMDA modulator Acamprosate calcium Chemical Structure
  33. GC62829 Afizagabar Afizagabar (S44819) is a first-in-class, competitive, and selective antagonist at the GABA-binding site of the α5-GABAAR, with an IC50 of 585 nM for α5β2γ2 and a Ki of 66 nM for α5β3γ2. Afizagabar Chemical Structure
  34. GC30844 Afloqualone An Analytical Reference Standard Afloqualone Chemical Structure
  35. GC14192 Allopregnanolone Allopregnanolone, a 3alpha, 5alpha progesterone metabolite, acts as a potent allosteric modulator of the γ-aminobutyric acid type A (GABAA) receptor, exerts antidepressant and neuroprotective action. Allopregnanolone Chemical Structure
  36. GC63495 Alogabat Alogabat (example 8) is a GABAA α5 receptor positive allosteric modulators (PAMs) (extracted from patent WO2018104419A1). Alogabat Chemical Structure
  37. GC30983 alpha-Asarone (α-Asarone) alpha-Asarone (α-Asarone) (α-Asarone) is one of the main psychoactive compounds, and possesses an antidepressant-like activity in mice. alpha-Asarone (α-Asarone) Chemical Structure
  38. GC13515 Alphaxalone activates and potentiates GABAA receptor-activated membrane current (IGABA) Alphaxalone Chemical Structure
  39. GC34064 Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) Aminooxyacetic acid (Carboxymethoxylamine) hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T. Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) Chemical Structure
  40. GC60596 Arecaidine Arecaidine, a pyridine alkaloid, is a potent GABA uptake inhibitor. Arecaidine Chemical Structure
  41. GC63879 Arecaidine hydrochloride Arecaidine hydrochloride, a pyridine alkaloid, is a potent GABA uptake inhibitor. Arecaidine hydrochloride Chemical Structure
  42. GC10974 AWD 131-138 AWD 131-138 (AWD 131-138) is a new low-affinity partial benzodiazepine receptor agonist with potent anticonvulsant and anxiolytic properties in rodent models. AWD 131-138 Chemical Structure
  43. GC31010 AZD-6280 AZD-6280 is a selective GABAA(α2/3) receptor modulator, used for treatment of generalized anxiety disorder. AZD-6280 Chemical Structure
  44. GC31990 Bamaluzole Bamaluzole is a GABA receptor agonist extracted from patent WO 2012064642 A1. Bamaluzole Chemical Structure
  45. GC19057 Basmisanil Basmisanil is a highly selective GABAAα5 negative allosteric modulator. Basmisanil Chemical Structure
  46. GC12414 Bemegride GABA receptor antagonist Bemegride Chemical Structure
  47. GC34494 Bifenazate An acaricide Bifenazate Chemical Structure
  48. GC11565 Bretazenil GABAA benzodiazepine site partial agonist Bretazenil Chemical Structure
  49. GC30521 Broflanilide Broflanilide is a potential insecticide and metabolized to Desmethyl-Broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin (RDL) GABA Receptor, and inhibits S. Broflanilide Chemical Structure
  50. GC31224 Carburazepam (RGH 3331) Carburazepam (RGH 3331) is a drug which derives from benzodiazepine. Carburazepam (RGH 3331) Chemical Structure
  51. GC13374 CGP 13501 Positive modulator of GABAB receptors,allosteric CGP 13501 Chemical Structure
  52. GC11153 CGP 35348 Selective GABAB antagonist, brain penetrant CGP 35348 Chemical Structure
  53. GC13676 CGP 36216 hydrochloride Selective GABAB antagonist CGP 36216 hydrochloride Chemical Structure
  54. GC35669 CGP 36742 CGP 36742 is a selective GABAB receptor antagonist that can penetrate the blood–brain barrier after peripheral administration, with an IC50 of 32?μM. CGP 36742 Chemical Structure
  55. GC13131 CGP 46381 GABAB receptor antagonist CGP 46381 Chemical Structure
  56. GC16947 CGP 52432 GABAB receptor antagonist CGP 52432 Chemical Structure
  57. GC10489 CGP 54626 hydrochloride

    GABAB receptor antagonist

     CGP 54626 hydrochloride Chemical Structure
  58. GC16600 CGP 55845 hydrochloride GABAB receptor antagonist CGP 55845 hydrochloride Chemical Structure
  59. GC15563 CGP 7930 Positive allosteric modulator of GABAB receptors CGP 7930 Chemical Structure
  60. GC33751 CGP11952 CGP11952 is a triazolyl-Benzaphenon resembling the benzodiazepines in its pharmacological action. CGP11952 Chemical Structure
  61. GC14274 CGS 20625 partial agonist for the benzodiazepine binding site of the GABAA receptor CGS 20625 Chemical Structure
  62. GC16311 Chlormethiazole hydrochloride GABAA agonist Chlormethiazole hydrochloride Chemical Structure
  63. GC16691 Chlormezanone Anxiolytic and skeletal muscle relaxant Chlormezanone Chemical Structure
  64. GC43261 Cholesteryl Myristate Cholesteryl Myristate is a natural steroid present in traditional Chinese medicine. Cholesteryl Myristate binds to several ion channels such as the nicotinic acetylcholine receptor, GABAA receptor, and the inward-rectifier potassium ion channel. Cholesteryl Myristate Chemical Structure
  65. GC14477 CI 966 hydrochloride GABA transporter GAT-1 inhibitor CI 966 hydrochloride Chemical Structure
  66. GC31120 Cirsimaritin Cirsimaritin binds weakly to the benzodiazepine site on GABAA receptors, with antidepressant, anxiolytic and antinociceptive activities. Cirsimaritin Chemical Structure
  67. GC16188 CL 218872 Benzodiazepine agonist CL 218872 Chemical Structure
  68. GC38758 Clomethiazole Chlormethiazole is an potent and orally active GABAA?agonist. Clomethiazole Chemical Structure
  69. GC60723 COR659 COR659 is a potent and effective GABAB positive allosteric modulator (PAM). COR659 Chemical Structure
  70. GC31052 CP-409092 CP-409092 is a partial agonist of GABAA receptor, with anti-anxiety activity. CP-409092 Chemical Structure
  71. GC38387 CP-409092 hydrochloride CP-409092 hydrochloride is a partial agonist of GABAA receptor, with anti-anxiety activity. CP-409092 hydrochloride Chemical Structure
  72. GC30930 DAA-1106 A TSPO agonist DAA-1106 Chemical Structure
  73. GC10530 Dihydroergotoxine mesylate GABAA receptor modulator Dihydroergotoxine mesylate Chemical Structure
  74. GC13405 DMCM hydrochloride Benzodiazepine inverse agonist DMCM hydrochloride Chemical Structure
  75. GC63590 Doxefazepam Doxefazepam Chemical Structure
  76. GC14150 DPNI-caged-GABA

    activates GABAA receptor

     DPNI-caged-GABA Chemical Structure
  77. GC12008 DS2 Positive allosteric modulator of δ-subunit containing GABAA receptors DS2 Chemical Structure
  78. GC35975 Emamectin Benzoate Emamectin Benzoate (MK-244) is an orally active nervoussystem toxicant by binding g-aminobutyric (GABA) receptor in insects. Emamectin Benzoate Chemical Structure
  79. GC11054 Epiallopregnanolone inactive as a GABAA receptor modulator and used as a control substance to examine GABA neurotransmission. Epiallopregnanolone Chemical Structure
  80. GC64673 Etbicyphat Etbicyphat (Trimethylopropane phosphate) is a potent GABA(A) receptors competitive antagonist. Etbicyphat Chemical Structure
  81. GC31023 Ethyl dirazepate Ethyl dirazepate is a drug which is a benzodiazepine derivative. Ethyl dirazepate Chemical Structure
  82. GC36012 Etifoxine A positive allosteric modulator of GABAA receptors Etifoxine Chemical Structure
  83. GC15264 Etifoxine hydrochloride A positive allosteric modulator of GABAA receptors Etifoxine hydrochloride Chemical Structure
  84. GC61788 Etiocholanolone An androgenically inactive metabolite of testosterone and androstenedione Etiocholanolone Chemical Structure
  85. GC16134 Etomidate

    General anesthetic with GABA modulatory and GABA-mimetic actions

     Etomidate Chemical Structure
  86. GC16985 Etomidate hydrochloride

    GABAA receptors agonist

     Etomidate hydrochloride Chemical Structure
  87. GC12568 FG 7142 benzodiazepine inverse agonist and anxiogenic agent FG 7142 Chemical Structure
  88. GC33754 FG8119 (NNC13-8119) FG8119 (NNC13-8119) is a novel benzodiazepine agonist extracted from patent US 4745112 A. FG8119 (NNC13-8119) Chemical Structure
  89. GC14017 FGIN-1-27

    high affinity agonist of the translocator protein (TSPO,peripheral benzodiazepine receptor)

     FGIN-1-27 Chemical Structure
  90. GC16238 FGIN-1-43 ligand as probe for the mitochondial DBI receptor (peripheral benzodiazepine receptor) FGIN-1-43 Chemical Structure
  91. GC60167 Fipronil An insecticide Fipronil Chemical Structure
  92. GC10772 Flumazenil

    Benzodiazepine antagonist

     Flumazenil Chemical Structure
  93. GC36058 Flumazenil acid Flumazenil acid is a metabolite of Flumazenil. Flumazenil acid Chemical Structure
  94. GC30088 Fluxametamide Fluxametamide is an insecticide with wide spectrum, acts as an antagonist of GABA- and glutamate-gated chloride channels, with IC50 of 1.95 nM and 225 nM for M. Fluxametamide Chemical Structure
  95. GC60862 GABAA receptor agent 1 GABAA receptor agent 1 is a high affinity ligand for GABAA receptor, with potent anticonvulsant activity. GABAA receptor agent 1 Chemical Structure
  96. GC12714 Gabapentin

    GABA enhancer

     Gabapentin Chemical Structure
  97. GC38543 Gaboxadol hydrochloride A GABAA receptor agonist and GABAC receptor antagonist Gaboxadol hydrochloride Chemical Structure
  98. GC11156 Ganaxolone positive allosteric modulator of GABAA receptor Ganaxolone Chemical Structure
  99. GC16495 GBLD 345 GABAA receptor agonist GBLD 345 Chemical Structure
  100. GC69161 Gidazepam

    Gidazepam is a GABA receptor channel (GABA RCs) agonist.

     Gidazepam Chemical Structure
  101. GC31205 Gidazepam (Gidasepam)

    Gidazepam is an agonist of GABA receptor channels (GABA RCs).

     Gidazepam (Gidasepam) Chemical Structure

Items 1 to 100 of 211 total

per page
  1. 1
  2. 2
  3. 3

Set Descending Direction