Others

CMKLR1 antagonist 1 (compound S-26d) is a potent and orally active chemokine-like receptor 1 (CMKLR1) antagonist, with a pIC50 value of 7.44 in hCMKLR1-transfected CHO cells.

RNF114 ligand 1 is a E3 Ubiquitin ligase binder.

5-PT formic is a serotonin derivative that can be functionalized with various reporter groups via click chemistry to investigate protein serotonylation.

Bexicaserin (Compound 3) is a 5-HT2C receptor agonist with potential for studying obesity and psychiatric-related diseases.

Orziloben is a medium chain fatty acid (MCFA) analogue.

2-Quinizarincarboxylic acid (Compound 15) is a glucose uptake inhibitor, with the inhibitory rate of 24.9% at 50 μM.

hRIO2 kinase ligand-1 (com 9) is a ligand of hRIO2 kinase, with a Kd value of 520 nM.

TNIK-IN-6 (Compound 9) is an inhibitor of Traf2 and Nck-interacting kinase (TNIK) and , with IC50 of 0.93 μM, that plays important roles in neurological and psychiatric disorders.

MMH1 is a novel BRD4 molecular glue degrader that functions by recruiting the CUL4 and DCAF16 ligases to the second bromodomain of BRD4 (BRD4BD2).

MMH2 is a novel BRD4 molecular glue degrader that functions by recruiting the CUL4 and DCAF16 ligases to the second bromodomain of BRD4 (BRD4BD2).

MNG-14a is an amphiphilic compound that can be used to aid the isolation of membrane proteins, and functional and structural determination of membrane proteins.

BFF-816 is an orally active kynurenine aminotransferase II (KAT II) inhibitor.

NOX-6-18 (GPR132 antagonist 1) is a potent and highly selective antagonist of the G protein-coupled receptor GPR132 (IC₅₀ = 17nM).

ANAT inhibitor-4 tetralithium (compound BA2) is potent N-acetyltransferase (ANAT) inhibitor with a Ki value of 48 nM.

Azide-A-DSBSO crosslinker is a mass spectrometry (MS)-cleavable, membrane-permeable, homobifunctional, azide-labeled, acid-cleavable cross-linked peptide.

COP1-ATGL modulator 1 (86) is an orally active modulator for COP1-ATGL axis.

MMH1-NR, containing a non-reactive (ethyl) group is a negative control of MMH1.

MZ-101 is a glycogen synthase 1 (GYS1) inhibitor.

Cholesteryl-Teg azide is a cholesterol azide used for bioconjugation and oligonucleotide (RNA, etc.) modification.

Perforin-IN-2 is a benzosulfonamide perforin inhibitor that alleviates transplant rejection during allogeneic bone marrow/stem cell transplantation.

QL47R is an approximately isosteric analogue of QL47 .

Ceramide 3B is a ceramide 3 lipid class with aggregation behavior.

PSAR18-COOH is a derivative of PSAR extracted from patent WO2009064913A1.

rel-VU6021625 is the less active relative configuration of VU6021625 .