Others

(R)-DZD1516 is the R enantiomer of DZD1516.

hCES2-IN-1 (Compound 24) is a reversible and selective hCES2 inhibitor (IC50: 6.72 μM).

FLT3/CHK-IN-1 (Compound 18) is a dual inhibitor of FLT3/CHK1.

Anticancer agent 168 (compound d16) is a inhibitor of DNA2.

PSMA-BCH (NOTA-PSMA) is a NOTA-conjugated precursor.

BLK degrader 1 (compound 9) is a selective degrader of B-lymphoid tyrosine kinase (BLK).

droxy-PP is a potent CBR1 inhibitor with an IC50 value of 0.78 μM. droxy-PP also potently inhibits the cytoplasmic tyrosine kinase Fyn with an IC50 value of 5 nM.

nti-inflammatory agent 49 (compound SC9) is a quite potent and selective inhibitor of Drp1-Fis1 interaction and can reduce FIS1-mediated mitochondrial dysfunction.

DQP-997-74 (compound 2i) is a selective inhibitor of N-metl-d-aspartate receptor (NMDAR), specifically targeting GluN2C/D (IC50: 0.069 μM and 0.035 μM), with blood-brain barrier penetrability.

Antiproliferative agent-37 (compound 10J) shows anti-proliferative effect by arresting the cells at the G2/M phase of the cell cycle.

NR2F2-IN-1 (free base) is a potent and selective orphan nuclear receptor COUP-TFII (NR2F2) inhibitor.

RGB-1 is a polycyclic aromatic drocarbon molecule and a stabilizer of RNA G-quadruplexes.

MN551 is a potent inhibitor of cysteine-directed electrophilic covalent that plays important roles in the biology of SOCS2 and its CRL5 complex.

TT-012 specifically binds to dynamic MITF and destroys the latter's dimer formation and DNA-binding ability.

TINK-IN-1 (Compound 9) is a potent and selective Traf2- and Nck-interacting kinase (TNIK) inhibitor with an IC50 of 8 nM.

Rezatapopt is an antineoplastic agent, used to inhibit solid tumor with p53 mutation.

Tegomil fumarate is an immunomodulator.

Plecstatin-1 drochloride is an anticancer agent containing organoeuropium.

(S)-STX-478 is the S-enantiomer of STX-478.

NorA-IN-1 (Compound 16) is a NorA inhibitor.

Idasanutlin enantiomer is the isomer of Idasanutlin , and can be used as an experimental control.

Antitumor agent-119 (compound 13K) is a 2-benzoxazolyl drazone derivative with anticancer activities.

Antiproliferative agent-36 (compound 8i) is a benzothiazolyl drazones derived compound with antiproliferative activity.

Antitumor agent-120 (compound 1) is a flavonoid compound isolated from Kudzu root.