Membrane Transporter/Ion Channel
- Piezo Channels(1)
- Aquaporins(1)
- AMPAR(62)
- ATPase(83)
- Calcium Channel(316)
- Cannabinoid Transporters(6)
- CFTR(41)
- Chloride Channels(13)
- GABA Receptor(196)
- Gardos Channel(1)
- Glucose Transporters(9)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(21)
- Kv1.3(1)
- ICB(3)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(4)
- Monoamine transporter(17)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(18)
- NKCC(7)
- NMDA Receptor(83)
- Nucleoside Transporters(4)
- Pannexin-1(4)
- P2X purinergic receptor(73)
- P-gp(14)
- Proton Pump(55)
- Potassium Channel(283)
- Sodium Channel(189)
- TRP Channel(157)
- TRPV1(11)
- URAT1(8)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(25)
- CRAC Channel(14)
- EAAT2(6)
- HCN Channel(5)
- Na+/HCO3- Cotransporter(2)
- Na+/K+ ATPase(34)
- P-glycoprotein(57)
- iGluR(166)
- nAChR(99)
- VDAC(2)
- GlyR(1)
Products for Membrane Transporter/Ion Channel
- Cat.No. Product Name Information
- GC16823 Enniatin Complex ionophore
- GC18105 Enterostatin Enterostatin, human, mouse, rat is a pentapeptide that reduces fat intake.
- GC43623 Erastin2 Erastin2 is a potent system xc- inhibitor and ferroptosis-inducing agent [1].
- GC13809 Eslicarbazepine acetate antiepileptic drug
- GC48984 Esomeprazole An H+/K+-ATPase inhibitor
- GC14313 Esomeprazole Magnesium Proton pump inhibitor
- GC36009 Esomeprazole magnesium salt Esomeprazole magnesium salt ((S)-Omeprazole magnesium salt) is a potent and orally active proton pump inhibitor and reduces acid secretion through inhibition of the H+, K+-ATPase in gastric parietal cells.
- GC13022 Esomeprazole Magnesium trihydrate An H+/K+-ATPase inhibitor
- GC33575 Esomeprazole potassium salt ((S)-Omeprazole potassium) Esomeprazole potassium salt ((S)-Omeprazole potassium) ((S)-Omeprazole potassium salt) is a potent and orally active proton pump inhibitor and reduces acid secretion through inhibition of the H+, K+-ATPase in gastric parietal cells.
- GC10599 Esomeprazole Sodium Proton pump inhibitor
- GC48979 Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate) A substrate of multidrug resistance protein 2
- GC10964 Estradiol 17-(β-D-Glucuronide) (sodium salt) Estradiol 17-(β-D-Glucuronide) sodium, a metabolite of estrogen, is well known to cause intrahepatic cholestasis in humans.
- GC17065 Estradiol 3-(β-D-Glucuronide) (sodium salt) substrate for multidrug resistance protein 2 (MRP2)
- GC64673 Etbicyphat Etbicyphat (Trimethylopropane phosphate) is a potent GABA(A) receptors competitive antagonist.
- GC25386 Ethacrynate Sodium Ethacrynate Sodium (ethacrynic acid sodium) is the sodium salt form of ethacrynic acid, which inhibits symport of sodium, potassium, and chloride primarily in the ascending limb of Henle, but also in the proximal and distal tubules.
- GC14041 Ethacrynic Acid Na+/K+/2Cl- cotransporter NKCC2 inhibitor
- GC10519 Ethacrynic acid - d5 Used as an internal standard for GC- or LC-mass spectrometry
- GC33695 Ethosuximide An anticonvulsant
- GC15824 Ethyl 3-Aminobenzoate (methanesulfonate) Ethyl 3-Aminobenzoate (methanesulfonate) (MS-222) is common used to immobilize fish for marking or transport and to suppress sensory systems during invasive procedures.
- GC31023 Ethyl dirazepate Ethyl dirazepate is a drug which is a benzodiazepine derivative.
- GC36012 Etifoxine A positive allosteric modulator of GABAA receptors
- GC33700 Etiracetam (UCB 6474) Etiracetam (UCB 6474) (UCB 6474) is an acetylcholine agonist and a nootropic drug of the racetam family.
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GC16134
Etomidate
General anesthetic with GABA modulatory and GABA-mimetic actions
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GC16985
Etomidate hydrochloride
GABAA receptors agonist
- GC65248 Etripamil Etripamil (MSP-2017) is a short-acting L-type calcium-channel antagonist, can be used for the research of Paroxysmal Supraventricular Tachycardia (PSVT).
- GC30910 Eucalyptol (1,8-Cineole) A bicyclic monoterpene with diverse biological activities
- GC13947 Evans Blue tetrasodium salt Evans Blue tetrasodium salt is a potent inhibitor of L-glutamate uptake via the membrane bound excitatory amino acid transporter (EAAT).
- GC38389 Evenamide Evenamide (NW-3509) is an orally available voltage-gated sodium channel (VGSC) blocker (Ki=0.4 ?M) for the research of schizophrenia.
- GC66016 Evifacotrep Evifacotrep, a short transient receptor potential channel 5 (TRPC5) antagonist (WO2020061162, compound 100), can be used for the research of neurological diseases.
- GC25405 Evodine Evodine, a natural product extracted from Evodiae fructus (EF), is a biomarker for quality assessment of EF in the Chinese Pharmacopoeia. Evodine is a potent P-gp inhibitor.
- GC15941 EVP-6124 A partial agonist of α7 subunit-containing nAChRs
- GC11091 EVP-6124 hydrochloride A partial agonist of α7 subunit-containing nAChRs
- GC67895 EVT-401
- GC39748 Facinicline hydrochloride Facinicline hydrochloride (RG3487 hydrochloride) is an orally active nicotinic α7 receptor partial agonist, with a Ki of 6 nM for α7 human nAChR.
- GC36027 Fanapanel hydrate Fanapanel hydrate (ZK200775 hydrate) is a highly selective AMPA/kainate antagonist with little activity against NMDA; have Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively.
- GC19152 Fantofarone Fantofarone is a highly potent Calcium Channel antagonist.
- GC18223 Farampator Farampator is a positive allosteric modulator of AMPA receptors that has an EC50 value greater than 32 uM for evoking glutamate currents in isolated pyramidal neurons.
- GC43654 Fasentin Fasentin is an inhibitor of glucose transport.
- GC13869 Fasudil Calcium antagonist
- GC14289 Fasudil (HA-1077) HCl Fasudil (HA-1077; AT877) Hydrochloride is a nonspecific RhoA/ROCK inhibitor and also has inhibitory effect on protein kinases, with an Ki of 0.33 μM for ROCK1, IC50s of 0.158 μM and 4.58 μM, 12.30 μM, 1.650 μM for ROCK2 and PKA, PKC, PKG, respectively. Fasudil (HA-1077) HCl is also a potent Ca2+ channel antagonist and vasodilator.
- GC36034 FD 12-9 FD 12-9 is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively. Anti-glioblastoma activity.
- GC10522 Felbamate antagonist at the NMDA-associated glycine binding site
- GC15363 Felbamate hydrate N-methyl-D-aspartate (NMDA) inhibitor
- GC17173 Felodipine Selective L-type Ca2+ channel blocker
- GC66436 FEMA 4809 FEMA 4809 is a TRPM8 receptor agonist (EC50=0.2 nM) for use as a cooling agent. TRPM8 is the ion channel responsible for the cool perception.
- GC60834 Fenamic acid Fenamic acid (N-Phenylanthranilic acid, NPAA) is an orally active chloride channel blocker.
- GC18086 Fendiline (hydrochloride) α2-adrenergic receptor antagonist
- GC47338 Fenoxycarb A non-neurotoxic carbamate insecticide
- GC49278 Fenpropathrin A pyrethroid insecticide
- GC60165 Ferulamide Ferulamide is a Ferulic acid derivative isolated from Portulaca oleracea L.
- GC18641 Ferutinin Ferutinin is a plant-derived ester of a sesquiterpenic alcohol that acts as an agonist for estrogen receptor (ER) α (IC50 = 33.1 nM) and an agonist/antagonist for ERβ (IC50 = 180.5 nM).
- GC50649 FFN 200 dihydrochloride
- GC12568 FG 7142 benzodiazepine inverse agonist and anxiogenic agent
- GC33754 FG8119 (NNC13-8119) FG8119 (NNC13-8119) is a novel benzodiazepine agonist extracted from patent US 4745112 A.
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GC14017
FGIN-1-27
high affinity agonist of the translocator protein (TSPO,peripheral benzodiazepine receptor)
- GC16238 FGIN-1-43 ligand as probe for the mitochondial DBI receptor (peripheral benzodiazepine receptor)
- GC63444 Filapixant Filapixant is a purinoreceptor antagonist extracted from patent WO2016091776A1, example 348.
- GC47352 FK-506-13C-d2 An internal standard for the quantification of FK-506
- GC49102 Flavoxate-d5 An internal standard for the quantification of flavoxate
- GC65416 Flecainide Flecainide is a potent and orally active antiarrhythmic agent.
- GC15823 Flecainide acetate An inhibitor of cardiac late sodium current
- GC65150 Flecainide hydrochloride Flecainide hydrochloride is a potent and orally active antiarrhythmic agent.
- GC47354 Flonicamid A pyridinecarboxamide insecticide
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GC13466
Flufenamic acid
TRPC activator
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GC10772
Flumazenil
Benzodiazepine antagonist
- GC36058 Flumazenil acid Flumazenil acid is a metabolite of Flumazenil.
- GC16532 Flunarizine 2HCl Flunarizine 2HCl is a potent dual Na+/Ca2+ channel (T-type) blocker.
- GC49739 Fluo-2 (potassium salt) A cell-impermeable fluorescent calcium indicator
- GC49458 Fluo-2 AM A cell-permeable fluorescent calcium indicator
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GC43681
Fluo-3 (ammonium salt)
Fluo-3 (ammonium salt) is a fluorescent calcium indicator commonly used in flow cytometry and cell-based experiments to detect changes in intracellular calcium levels.
- GC43682 Fluo-3 (potassium salt) Fluo-3 (potassium salt) is a fluorescent calcium indicator commonly used in flow cytometry and cell-based experiments to detect changes in intracellular calcium levels.
- GC43683 Fluo-3 (sodium salt) Fluo-3 is a fluorescent calcium indicator commonly used in flow cytometry and cell-based experiments to detect changes in intracellular calcium levels.
- GC43684 Fluo-3FF (potassium salt) Fluo-3FF is a fluorescent calcium indicator.
- GC49741 Fluo-4 (potassium salt) A cell-impermeable fluorescent calcium indicator
- GC36060 Flupirtine Flupirtine(D 9998) is a selective neuronal potassium channel opener that also has NMDA receptor antagonist properties.
- GC11470 Flupirtine maleate NMDA receptor antagonist
- GC66073 Flupyradifurone Flupyradifurone is a systemic nAChR agonist that interferes with signal transduction in the central nervous system of sucking pests. Flupyradifurone can be used as a butenolide insecticide.
- GC64394 Flupyrimin Flupyrimin acts as an antagonist at the insect nicotinic acetylcholine receptor (nAChR).
- GC11492 Fluspirilene potent, non-competitive antagonist of agonist-activated L-type calcium channels
- GC49397 Fluvoxamine-d4 (maleate) An internal standard for the quantification of fluvoxamine
- GC30088 Fluxametamide Fluxametamide is an insecticide with wide spectrum, acts as an antagonist of GABA- and glutamate-gated chloride channels, with IC50 of 1.95 nM and 225 nM for M.
- GC10506 FPL 64176 L-type Ca2+ channels activator
- GC33895 FR183998 free base FR183998 free base is a potent Na+/H+-exchange inhibitor, with IC50s of 0.3 nM, 3.1 nM and 6.5 nM by measurement of pHi change in rat lymphocytes, rat and human platelets, respectively.
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GC49089
FR900359
A cyclic depsipeptide and an inhibitor of Gαq, Gα11, and Gα14
- GC18260 FTase Inhibitor I FTase inhibitor I is a potent inhibitor of farnesyltransferase (FTase; IC50 = 21 nM) that is greater than 30-fold selective for FTase over geranylgeranyl transferase (GGTase; IC50 = 790 nM).
- GC52503 FTase Inhibitor II (trifluoroacetate salt) A potent, selective inhibitor of farnesyltransferase
- GC10874 Fumitremorgin C multidrug transporter inhibitor
- GC30628 Funapide (TV 45070) Funapide (TV 45070) (TV 45070; XEN402) is a potent Sodium Channel Nav1.7 inhibitor.
- GC43711 Fura-2 (potassium salt) Fura-2 (potassium salt) is a scaled fluorescent dye that can be used for intracellular calcium imaging with the Kd value of 140 nM.
- GC43712 Fura-2 (sodium salt) Fura-2 is a ratiometric fluorescent calcium indicator that can be used to detect calcium in cells.
- GC49462 Fura-2 Leakage Resistant (potassium salt) A cell-impermeable, ratiometric fluorescent calcium indicator
- GC49465 Fura-2 Leakage Resistant AM A cell-permeable, ratiometric fluorescent calcium indicator
- GC43713 Fura-FF (potassium salt) Fura-FF (potassium salt) is a low-affinity fluorescent dye for calcium (Ex/Em: 365/514 nm in the absence of calcium; 339/507 nm in the presence of a high calcium concentration).
- GC43714 Fura-FF AM Fura-FF AM is a cell-permeable acetoxymethyl ester of the fluorescence calcium indicator fura-FF (potassium salt).
- GC12970 Furosemide GABAA receptors antagonist
- GC36091 Furosemide sodium A loop diuretic inhibitor of Na+/2Cl-/K+ (NKCC) cotransporter
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GC12714
Gabapentin
GABA enhancer
- GC36097 Gabapentin enacarbil Gabapentin enacarbil (XP-13512) is a prodrug for the anticonvulsant and analgesic drug gabapentin.
- GC17316 Gabapentin HCl Gabapentin HCl is a potent, orally active P/Q type Ca2+ channel blocker.
- GC38543 Gaboxadol hydrochloride A GABAA receptor agonist and GABAC receptor antagonist