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Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein

Products for  GPCR/G protein

  1. Cat.No. Product Name Information
  2. GC19077 BMS-813160 BMS-813160 is the first dual CCR2/CCR5 antagonist to enter clinical development for cardiovascular. BMS-813160 Chemical Structure
  3. GC31479 BMS-819881 BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM. BMS-819881 Chemical Structure
  4. GC19078 BMS-986020 BMS-986020 is an LPA1 antagonist. BMS-986020 Chemical Structure
  5. GC38470 BMS-986020 sodium BMS-986020 (AM152) sodium is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist. BMS-986020 sodium Chemical Structure
  6. GC63895 BMS-986278 BMS-986278 is a potent lysophosphatidic acid receptor 1 (LPA1) antagonist, with a human LPA1 Kb of 6.9 nM. BMS-986278 Chemical Structure
  7. GC31081 BMT-145027 BMT-145027 is an mGluR5 positive allosteric modulator without inherent agonist activity, exhibits an EC50 of 47 nM. BMT-145027 Chemical Structure
  8. GC13796 BMY 14802 hydrochloride Sigma receptor antagonist BMY 14802 hydrochloride Chemical Structure
  9. GC11820 BMY 45778 partial agonist at IP1 prostacyclin receptors BMY 45778 Chemical Structure
  10. GC10848 BMY 7378 5-HT1A partial agonist and α1D adrenoceptor antagonist BMY 7378 Chemical Structure
  11. GC11278 Boc-MLF formyl peptide receptor 1 (FPR1) antagonist Boc-MLF Chemical Structure
  12. GC14014 Bombesin Neuropeptide with many biological effects Bombesin Chemical Structure
  13. GC16761 Bombinakinin M Potent bradykinin receptor agonist Bombinakinin M Chemical Structure
  14. GC14629 Bombinakinin-GAP Bioactive bradykinin-related peptide Bombinakinin-GAP Chemical Structure
  15. GC32665 Bometolol Hydrochloride Bometolol Hydrochloride is a beta-adrenergic blocking agent, used for the research of cardiovascular disease. Bometolol Hydrochloride Chemical Structure
  16. GC16269 Bosentan Endothelin receptor antagonist Bosentan Chemical Structure
  17. GC11465 Bosentan Hydrate endothelin receptor antagonist Bosentan Hydrate Chemical Structure
  18. GC19081 BPTU BPTU is a novel P2Y1 allosteric antagonist. BPTU Chemical Structure
  19. GC15887 BQ-123 Selective ETA receptor antagonist BQ-123 Chemical Structure
  20. GC14416 BQ-3020 ETB receptor agonist,potent and selective BQ-3020 Chemical Structure
  21. GC60094 BQ-3020 TFA BQ-3020 (TFA) is a selective agonist of ETB receptor, inhibits [125I]ET-1 binding to ETB receptor with an IC50 of 0.2 nM in cerebellum, and causes vasoconstriction. BQ-3020 TFA Chemical Structure
  22. GC35546 BQ-788 BQ-788 is a potent, selective ETB receptor antagonist with IC50 of 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells, poorly inhibiting the binding to ETA receptors in human neuroblastoma cell line SK-N-MC cells with IC50 of 1300 nM. BQ-788 Chemical Structure
  23. GC15916 BQ-788 sodium salt ET B-receptor antagonist,potent and selective BQ-788 sodium salt Chemical Structure
  24. GC15758 BQCA positive allosteric modulator of the M1 muscarinic acetylcholine receptor (mAChR) BQCA Chemical Structure
  25. GC10612 BQU57 Derivative of RBC8 BQU57 Chemical Structure
  26. GC35548 Bradykinin Bradykinin is an active peptide that is generated by the kallikrein-kinin system. Bradykinin Chemical Structure
  27. GC32576 Bradykinin 1-3 Bradykinin 1-3 is a 3-amino acid residue peptide. Bradykinin 1-3 Chemical Structure
  28. GC32592 Bradykinin 1-5 Bradykinin 1-5 is a major stable metabolite of Bradykinin, formed by the proteolytic action of angiotensin-converting enzyme (ACE). Bradykinin 1-5 Chemical Structure
  29. GC32605 Bradykinin 1-6 Bradykinin 1-6 is an amino-truncated Bradykinin peptide. Bradykinin 1-6 Chemical Structure
  30. GC32601 Bradykinin 1-7(Bradykinin Fragment 1-​7) Bradykinin 1-7 (Bradykinin Fragment 1-​7) is an amino-truncated Bradykinin peptide. Bradykinin 1-7(Bradykinin Fragment 1-​7) Chemical Structure
  31. GC34042 Bradykinin 2-9 (Des-Arg1-bradykinin) Bradykinin 2-9 (Des-Arg1-bradykinin) is an amino-truncated Bradykinin peptide. Bradykinin 2-9 (Des-Arg1-bradykinin) Chemical Structure
  32. GC60095 Brain Natriuretic Peptide (1-32), rat acetate Brain Natriuretic Peptide (1-32), rat acetate (BNP (1-32), rat acetate) is a 32 amino acid polypeptide secreted by the ventricles of the heart in response to excessive stretching of heart muscle cells (cardiomyocytes). Brain Natriuretic Peptide (1-32), rat acetate Chemical Structure
  33. GC32589 Brain Natriuretic Peptide (BNP) (1-32), rat Brain Natriuretic Peptide (BNP) (1-32), rat (BNP (1-32), rat) is a 32 amino acid polypeptide secreted by the ventricles of the heart in response to excessive stretching of heart muscle cells (cardiomyocytes). Brain Natriuretic Peptide (BNP) (1-32), rat Chemical Structure
  34. GC34002 Bremelanotide Acetate (PT-141 Acetate) Bremelanotide Acetate (PT-141 Acetate) (PT-141 Acetate), a synthetic peptide analogue of α-MSH, is an agonist at melanocortin receptors including the MC3R and MC4R for the treatment of sexual dysfunction. Bremelanotide Acetate (PT-141 Acetate) Chemical Structure
  35. GC11186 Brexpiprazole 5-HT2A, α1B-, and α2C-adrenergic receptors antagonist Brexpiprazole Chemical Structure
  36. GC10738 Brimonidine Tartrate Highly selective α-adrenergic receptor agonist Brimonidine Tartrate Chemical Structure
  37. GC13785 BRL 37344, sodium salt BRL 37344, sodium salt (BRL 37344A) is a specific β3-adrenergic receptor agonist. BRL 37344, sodium salt Chemical Structure
  38. GC13996 BRL 44408 maleate Selective α2A-AR antagonist BRL 44408 maleate Chemical Structure
  39. GC16226 BRL-15572 dihydrochloride BRL-15572 is a selective antagonist of h5-HT1D, displays high affinity for h5-HT1D receptors. BRL-15572 dihydrochloride Chemical Structure
  40. GC17130 BRL-54443 5-HT1E/1F receptor agonist,potent and selective BRL-54443 Chemical Structure
  41. GC30989 Bromperidol (R-11333) Bromperidol (R-11333) (R-11333) possesses antipsychotic activity, with a high affinity for central dopamine receptors D2. Bromperidol (R-11333) Chemical Structure
  42. GC32039 BTM-1086 BTM-1086 is a potent anti-ulcer and gastric secretory inhibiting agent. BTM-1086 Chemical Structure
  43. GC15328 Bucindolol beta adrenergic blocker Bucindolol Chemical Structure
  44. GC11897 Budesonide Anti-inflammatory corticosteroid Budesonide Chemical Structure
  45. GC67692 Bufuralol Bufuralol Chemical Structure
  46. GC15347 Bufuralol (hydrochloride) non-specific β-adrenergic blocker Bufuralol (hydrochloride) Chemical Structure
  47. GC32002 Bunaprolast (U66858) Bunaprolast (U66858) (U66858) is a potent inhibitor of LTB4 production in human whole blood. Bunaprolast (U66858) Chemical Structure
  48. GC64450 Bunazosin Bunazosin is a potent and selective α1-adrenoceptor antagonist. Bunazosin Chemical Structure
  49. GC62648 Bupranolol Bupranolol is an orally active, competitive and non-selective β-adrenoceptor antagonist without intrinsic sympathomimetic activity. Bupranolol Chemical Structure
  50. GC30625 Burixafor hydrobromide (TG-0054 hydrobromide) Burixafor hydrobromide (TG-0054 hydrobromide) (TG-0054 hydrobromide) is an orally bioavailable and potent antagonist of CXCR4 and a well anti-angiogenic drug that is of potential value in treating choroid neovascularization. Burixafor hydrobromide (TG-0054 hydrobromide) Chemical Structure
  51. GC11191 Buspirone HCl Buspirone HCl is a 5-HT1A receptor agonist. Buspirone HCl Chemical Structure
  52. GC16539 Butaprost A selective agonist for the EP2 receptors Butaprost Chemical Structure
  53. GC11584 Butenoyl PAF PAF receptor agonist Butenoyl PAF Chemical Structure
  54. GC64504 Butyryltimolol Butyryltimolol, an effective prodrug of Timolol, improves the corneal penetration of Timolol. Butyryltimolol Chemical Structure
  55. GC14393 BVD 10 NPY Y1 receptor antagonist,highly selective BVD 10 Chemical Structure
  56. GC14212 BW 245C DP1 receptor agonist BW 245C Chemical Structure
  57. GC14859 BW 246C DP receptor agonist BW 246C Chemical Structure
  58. GC11231 BW 723C86 hydrochloride BW 723C86 hydrochloride is a potent and a selective 5-HT2B receptor agonist. BW 723C86 hydrochloride Chemical Structure
  59. GC17348 BW A868C prostaglandin D2 antagonist BW A868C Chemical Structure
  60. GC14789 BWX 46 NPY Y5 receptor agonist,potent and highly selective BWX 46 Chemical Structure
  61. GC14519 BX 471 CCR1 antagonist,potent and selective BX 471 Chemical Structure
  62. GC13299 BX 513 hydrochloride Selective CCR1 antagonist BX 513 hydrochloride Chemical Structure
  63. GC35570 BX471 hydrochloride BX471 hydrochloride (ZK-811752 hydrochloride) is a potent, selective non-peptide CCR1 antagonist with Ki of 1 nM for human CCR1, and exhibits 250-fold selectivity for CCR1 over CCR2, CCR5 and CXCR4. BX471 hydrochloride Chemical Structure
  64. GC11161 C 021 dihydrochloride C 021 dihydrochloride is a potent CC chemokine receptor-4 (CCR4) antagonist. C 021 dihydrochloride Chemical Structure
  65. GC12034 C-type natriuretic peptide (1-22) (human, rat, swine) C-type natriuretic peptide (1-22) (human, rat, swine), a 1-22 fragment of CNP, is a natriuretic peptide receptor B (NPR-B) agonist. C-type natriuretic peptide (1-22) (human, rat, swine) Chemical Structure
  66. GC35756 C-Type Natriuretic Peptide (1-53), human C-Type Natriuretic Peptide (1-53), human is the 1-53 fragment of C-Type Natriuretic Peptide. C-Type Natriuretic Peptide (1-53), human Chemical Structure
  67. GC68908 C-Type Natriuretic Peptide (1-53), human TFA

    C-Type Natriuretic Peptide (1-53), human TFA is a fragment of C-type natriuretic peptide consisting of amino acids 1 to 53. C-Type Natriuretic Peptide TFA belongs to the family of natriuretic peptides and is involved in maintaining electrolyte-fluid balance and vascular tone.

     C-Type Natriuretic Peptide (1-53), human TFA Chemical Structure
  68. GC17244 Calcium-Sensing Receptor Antagonists I Calcium-Sensing Receptor Antagonists I Chemical Structure
  69. GC17697 Calhex 231 hydrochloride

    negative allosteric modulator of Ca2+-sensing receptor (CaSR)

     Calhex 231 hydrochloride Chemical Structure
  70. GC12620 Calindol (hydrochloride) activator of the calcium-sensing receptor (CaSR) Calindol (hydrochloride) Chemical Structure
  71. GC65081 CALP1 TFA CALP1 TFA is a calmodulin (CaM) agonist (Kd of 88 ?M) with binding to the CaM EF-hand/Ca2+-binding site. CALP1 TFA Chemical Structure
  72. GC31072 Camylofine

    Camylofin is an antimuscarinic, is a smooth muscle relaxant

     Camylofine Chemical Structure
  73. GC16978 Candesartan Angiotensin II receptor 1 (AT1) antagonist Candesartan Chemical Structure
  74. GC12318 Candesartan Cilexetil Prodrug of the angiotensin II receptor 1 (AT1) antagonist candesartan Candesartan Cilexetil Chemical Structure
  75. GC40238 Candesartan-d4 Candesartan-d4 is intended for use as an internal standard for the quantification of candesartan by GC- or LC-MS. Candesartan-d4 Chemical Structure
  76. GC43137 Cangrelor (sodium salt) Cangrelor (sodium salt), an adenosine triphosphate analogue, is a reversible and selective platelet P2Y12 antagonist, with prompt and potent antiplatelet effects. Cangrelor (sodium salt) Chemical Structure
  77. GC14935 Capadenoson A partial adenosine receptor agonist Capadenoson Chemical Structure
  78. GC19087 Capromorelin Tartrate Capromorelin Tartrate is an orally active, potent growth hormone secretagogue receptor (GHSR) agonist, with Ki of 7 nM for hGHS-R1a. Capromorelin Tartrate Chemical Structure
  79. GC13180 Carazolol high-affinity, lipophilic, non-selective ligand of the β-adrenergic receptors Carazolol Chemical Structure
  80. GC32487 Carbacyclin (Carbaprostacyclin) Carbacyclin (Carbaprostacyclin) is a PGI2 analogue, acts as a prostacyclin (PGI2) receptor agonist and vasodilator, and potently inhibits platelet aggregation. Carbacyclin (Carbaprostacyclin) Chemical Structure
  81. GC16937 Carbamoylcholine chloride

    Cholinergic receptor agonist

     Carbamoylcholine chloride Chemical Structure
  82. GC15243 Carbazochrome sodium sulfonate (AC-17) Carbazochrome sodium sulfonate (AC-17) (AC-17) is a capillary stabiliser and used for the research of haemorrhage. Carbazochrome sodium sulfonate (AC-17) Chemical Structure
  83. GC11419 Carbetocin oxytocin receptor agonist Carbetocin Chemical Structure
  84. GC50450 Carboprost tromethamine Synthetic Prostaglandin F2α analog Carboprost tromethamine Chemical Structure
  85. GC35610 Cariprazine hydrochloride An atypical antipsychotic Cariprazine hydrochloride Chemical Structure
  86. GC46007 Cariprazine-d6 An internal standard for the quantification of cariprazine Cariprazine-d6 Chemical Structure
  87. GC68832 Carlumab

    Carlumab (CNTO 888) is a highly-affinity humanized antibody against CCL2 (chemokine ligand 2). Carlumab can be used for cancer research, especially in prostate cancer.

     Carlumab Chemical Structure
  88. GC17864 CART (55-102) (human) CART with potent appetite-suppressing activity CART (55-102) (human) Chemical Structure
  89. GC11131 CART (55-102) (rat) CART with potent appetite-suppressing activity CART (55-102) (rat) Chemical Structure
  90. GC14034 CART (62-76) (rat, human) CART (62-76) (rat, human) is a neuropeptide (62-76 residues of the CART peptide) with neurotransmitter-like effects. CART (62-76) (rat, human) Chemical Structure
  91. GC16395 Carteolol HCl Carteolol HCl (OPC-1085 hydrochloride) is a non-selective beta blocker used to treat glaucoma. Carteolol HCl Chemical Structure
  92. GC14769 Carvedilol Potent β-adrenoceptor and α1-adrenoceptor antagonist Carvedilol Chemical Structure
  93. GC25197 Carvedilol EP IMpurity E Carvedilol is a nonselective beta blocker/alpha-1 blocker and used in management of congestive heart failure (CHF). Carvedilol EP IMpurity E Chemical Structure
  94. GC35613 Carvedilol phosphate hemihydrate Carvedilol phosphate hemihydrate (BM 14190 phosphate hemihydrate) is a non-selective β/α-1 blocker. Carvedilol phosphate hemihydrate Chemical Structure
  95. GC64003 Carvedilol-d4 Carvedilol-d4 Chemical Structure
  96. GC16692 Casin GTPase Cdc42 inhibitor Casin Chemical Structure
  97. GC62888 Casopitant mesylate Casopitant mesylate (GW679769B) is a potent, selective, brain permeable and orally active neurokinin 1 (NK1) receptor antagonist. Casopitant mesylate Chemical Structure
  98. GC50293 CATPB FFA2 (GPR43) inverse agonist CATPB Chemical Structure
  99. GC18318 CAY10441 CAY10441 is a potent and selective IP (prostacyclin) receptor antagonist. CAY10441 Chemical Structure
  100. GC35620 CAY10471 Racemate CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist, with a Ki of 0.6 nM for hCRTH2, selective over human thromboxane A2 receptor TP (Ki, >10000 nM) or PGD2 receptor DP (Ki, 1200 nM). CAY10471 Racemate Chemical Structure
  101. GC18678 CAY10595 The biological effects of prostaglandin D2 (PGD2) are transduced by at least two 7-transmembrane G protein-coupled receptors, designated DP1 and CRTH2/DP2. CAY10595 Chemical Structure

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