GPCR/G protein
- Neuropeptide FF/AF Receptors(43)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(415)
- Acetylcholine(19)
- Adenosine Deaminase(12)
- Adenosine Receptor(133)
- Adenosine Kinase(5)
- Adiponectin Receptor(4)
- Adrenergic Receptor(404)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(110)
- Bombesin Receptors(22)
- Bradykinin Receptors(27)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(137)
- Calcimimetic Agent(3)
- CaSR(24)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(79)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(82)
- CysLT1 receptor(1)
- Endothelin Receptor(50)
- EP1 Receptor(3)
- EP4 Receptor(5)
- ERRγ(2)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(20)
- Galanin Receptors(11)
- Ghrelin Receptors(12)
- GHSR(22)
- GIP Receptor(5)
- Glucagon Receptor(66)
- Glucocorticoid Receptor(87)
- GLUT1(2)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(13)
- GPR109A(4)
- GPR119(11)
- GPR120(12)
- GPR35(8)
- GPR44(1)
- GPR55(10)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(55)
- LPA Receptor(15)
- LPL Receptor(60)
- LTD4 Receptor(2)
- mGluR (115)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(49)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(21)
- NK2 Receptors(7)
- NK3 Receptor(8)
- NOP Receptor(22)
- NPY Receptors(28)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(42)
- Oxytocin Receptors(21)
- P2Y Receptor(55)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(15)
- PGD2 Receptor(2)
- Prostaglandin Receptor(168)
- Prostanoid Receptors(25)
- Protease-Activated Receptors(10)
- RGS(4)
- S1P receptor(9)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(34)
- Sigma Receptor(54)
- Vasopressin Receptor(33)
- 17,20-lyase(7)
- Ras(118)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(5)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(22)
- GPR84(5)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(4)
- CRFR(21)
- RGS Protein(7)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(23)
- GPR139(3)
- mAChR(179)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(72)
- cGMP(18)
- GRK(1)
Products for GPCR/G protein
- Cat.No. Product Name Information
- GC19077 BMS-813160 BMS-813160 is the first dual CCR2/CCR5 antagonist to enter clinical development for cardiovascular.
- GC31479 BMS-819881 BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM.
- GC19078 BMS-986020 BMS-986020 is an LPA1 antagonist.
- GC38470 BMS-986020 sodium BMS-986020 (AM152) sodium is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist.
- GC63895 BMS-986278 BMS-986278 is a potent lysophosphatidic acid receptor 1 (LPA1) antagonist, with a human LPA1 Kb of 6.9 nM.
- GC31081 BMT-145027 BMT-145027 is an mGluR5 positive allosteric modulator without inherent agonist activity, exhibits an EC50 of 47 nM.
- GC13796 BMY 14802 hydrochloride Sigma receptor antagonist
- GC11820 BMY 45778 partial agonist at IP1 prostacyclin receptors
- GC10848 BMY 7378 5-HT1A partial agonist and α1D adrenoceptor antagonist
- GC11278 Boc-MLF formyl peptide receptor 1 (FPR1) antagonist
- GC14014 Bombesin Neuropeptide with many biological effects
- GC16761 Bombinakinin M Potent bradykinin receptor agonist
- GC14629 Bombinakinin-GAP Bioactive bradykinin-related peptide
- GC32665 Bometolol Hydrochloride Bometolol Hydrochloride is a beta-adrenergic blocking agent, used for the research of cardiovascular disease.
- GC16269 Bosentan Endothelin receptor antagonist
- GC11465 Bosentan Hydrate endothelin receptor antagonist
- GC19081 BPTU BPTU is a novel P2Y1 allosteric antagonist.
- GC15887 BQ-123 Selective ETA receptor antagonist
- GC14416 BQ-3020 ETB receptor agonist,potent and selective
- GC60094 BQ-3020 TFA BQ-3020 (TFA) is a selective agonist of ETB receptor, inhibits [125I]ET-1 binding to ETB receptor with an IC50 of 0.2 nM in cerebellum, and causes vasoconstriction.
- GC35546 BQ-788 BQ-788 is a potent, selective ETB receptor antagonist with IC50 of 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells, poorly inhibiting the binding to ETA receptors in human neuroblastoma cell line SK-N-MC cells with IC50 of 1300 nM.
- GC15916 BQ-788 sodium salt ET B-receptor antagonist,potent and selective
- GC15758 BQCA positive allosteric modulator of the M1 muscarinic acetylcholine receptor (mAChR)
- GC10612 BQU57 Derivative of RBC8
- GC35548 Bradykinin Bradykinin is an active peptide that is generated by the kallikrein-kinin system.
- GC32576 Bradykinin 1-3 Bradykinin 1-3 is a 3-amino acid residue peptide.
- GC32592 Bradykinin 1-5 Bradykinin 1-5 is a major stable metabolite of Bradykinin, formed by the proteolytic action of angiotensin-converting enzyme (ACE).
- GC32605 Bradykinin 1-6 Bradykinin 1-6 is an amino-truncated Bradykinin peptide.
- GC32601 Bradykinin 1-7(Bradykinin Fragment 1-7) Bradykinin 1-7 (Bradykinin Fragment 1-7) is an amino-truncated Bradykinin peptide.
- GC34042 Bradykinin 2-9 (Des-Arg1-bradykinin) Bradykinin 2-9 (Des-Arg1-bradykinin) is an amino-truncated Bradykinin peptide.
- GC60095 Brain Natriuretic Peptide (1-32), rat acetate Brain Natriuretic Peptide (1-32), rat acetate (BNP (1-32), rat acetate) is a 32 amino acid polypeptide secreted by the ventricles of the heart in response to excessive stretching of heart muscle cells (cardiomyocytes).
- GC32589 Brain Natriuretic Peptide (BNP) (1-32), rat Brain Natriuretic Peptide (BNP) (1-32), rat (BNP (1-32), rat) is a 32 amino acid polypeptide secreted by the ventricles of the heart in response to excessive stretching of heart muscle cells (cardiomyocytes).
- GC34002 Bremelanotide Acetate (PT-141 Acetate) Bremelanotide Acetate (PT-141 Acetate) (PT-141 Acetate), a synthetic peptide analogue of α-MSH, is an agonist at melanocortin receptors including the MC3R and MC4R for the treatment of sexual dysfunction.
- GC11186 Brexpiprazole 5-HT2A, α1B-, and α2C-adrenergic receptors antagonist
- GC10738 Brimonidine Tartrate Highly selective α-adrenergic receptor agonist
- GC13785 BRL 37344, sodium salt BRL 37344, sodium salt (BRL 37344A) is a specific β3-adrenergic receptor agonist.
- GC13996 BRL 44408 maleate Selective α2A-AR antagonist
- GC16226 BRL-15572 dihydrochloride BRL-15572 is a selective antagonist of h5-HT1D, displays high affinity for h5-HT1D receptors.
- GC17130 BRL-54443 5-HT1E/1F receptor agonist,potent and selective
- GC30989 Bromperidol (R-11333) Bromperidol (R-11333) (R-11333) possesses antipsychotic activity, with a high affinity for central dopamine receptors D2.
- GC32039 BTM-1086 BTM-1086 is a potent anti-ulcer and gastric secretory inhibiting agent.
- GC15328 Bucindolol beta adrenergic blocker
- GC11897 Budesonide Anti-inflammatory corticosteroid
- GC67692 Bufuralol
- GC15347 Bufuralol (hydrochloride) non-specific β-adrenergic blocker
- GC32002 Bunaprolast (U66858) Bunaprolast (U66858) (U66858) is a potent inhibitor of LTB4 production in human whole blood.
- GC64450 Bunazosin Bunazosin is a potent and selective α1-adrenoceptor antagonist.
- GC62648 Bupranolol Bupranolol is an orally active, competitive and non-selective β-adrenoceptor antagonist without intrinsic sympathomimetic activity.
- GC30625 Burixafor hydrobromide (TG-0054 hydrobromide) Burixafor hydrobromide (TG-0054 hydrobromide) (TG-0054 hydrobromide) is an orally bioavailable and potent antagonist of CXCR4 and a well anti-angiogenic drug that is of potential value in treating choroid neovascularization.
- GC11191 Buspirone HCl Buspirone HCl is a 5-HT1A receptor agonist.
- GC16539 Butaprost A selective agonist for the EP2 receptors
- GC11584 Butenoyl PAF PAF receptor agonist
- GC64504 Butyryltimolol Butyryltimolol, an effective prodrug of Timolol, improves the corneal penetration of Timolol.
- GC14393 BVD 10 NPY Y1 receptor antagonist,highly selective
- GC14212 BW 245C DP1 receptor agonist
- GC14859 BW 246C DP receptor agonist
- GC11231 BW 723C86 hydrochloride BW 723C86 hydrochloride is a potent and a selective 5-HT2B receptor agonist.
- GC17348 BW A868C prostaglandin D2 antagonist
- GC14789 BWX 46 NPY Y5 receptor agonist,potent and highly selective
- GC14519 BX 471 CCR1 antagonist,potent and selective
- GC13299 BX 513 hydrochloride Selective CCR1 antagonist
- GC35570 BX471 hydrochloride BX471 hydrochloride (ZK-811752 hydrochloride) is a potent, selective non-peptide CCR1 antagonist with Ki of 1 nM for human CCR1, and exhibits 250-fold selectivity for CCR1 over CCR2, CCR5 and CXCR4.
- GC11161 C 021 dihydrochloride C 021 dihydrochloride is a potent CC chemokine receptor-4 (CCR4) antagonist.
- GC12034 C-type natriuretic peptide (1-22) (human, rat, swine) C-type natriuretic peptide (1-22) (human, rat, swine), a 1-22 fragment of CNP, is a natriuretic peptide receptor B (NPR-B) agonist.
- GC35756 C-Type Natriuretic Peptide (1-53), human C-Type Natriuretic Peptide (1-53), human is the 1-53 fragment of C-Type Natriuretic Peptide.
-
GC68908
C-Type Natriuretic Peptide (1-53), human TFA
C-Type Natriuretic Peptide (1-53), human TFA is a fragment of C-type natriuretic peptide consisting of amino acids 1 to 53. C-Type Natriuretic Peptide TFA belongs to the family of natriuretic peptides and is involved in maintaining electrolyte-fluid balance and vascular tone.
- GC17244 Calcium-Sensing Receptor Antagonists I
-
GC17697
Calhex 231 hydrochloride
negative allosteric modulator of Ca2+-sensing receptor (CaSR)
- GC12620 Calindol (hydrochloride) activator of the calcium-sensing receptor (CaSR)
- GC65081 CALP1 TFA CALP1 TFA is a calmodulin (CaM) agonist (Kd of 88 ?M) with binding to the CaM EF-hand/Ca2+-binding site.
-
GC31072
Camylofine
Camylofin is an antimuscarinic, is a smooth muscle relaxant
- GC16978 Candesartan Angiotensin II receptor 1 (AT1) antagonist
- GC12318 Candesartan Cilexetil Prodrug of the angiotensin II receptor 1 (AT1) antagonist candesartan
- GC40238 Candesartan-d4 Candesartan-d4 is intended for use as an internal standard for the quantification of candesartan by GC- or LC-MS.
- GC43137 Cangrelor (sodium salt) Cangrelor (sodium salt), an adenosine triphosphate analogue, is a reversible and selective platelet P2Y12 antagonist, with prompt and potent antiplatelet effects.
- GC14935 Capadenoson A partial adenosine receptor agonist
- GC19087 Capromorelin Tartrate Capromorelin Tartrate is an orally active, potent growth hormone secretagogue receptor (GHSR) agonist, with Ki of 7 nM for hGHS-R1a.
- GC13180 Carazolol high-affinity, lipophilic, non-selective ligand of the β-adrenergic receptors
- GC32487 Carbacyclin (Carbaprostacyclin) Carbacyclin (Carbaprostacyclin) is a PGI2 analogue, acts as a prostacyclin (PGI2) receptor agonist and vasodilator, and potently inhibits platelet aggregation.
-
GC16937
Carbamoylcholine chloride
Cholinergic receptor agonist
- GC15243 Carbazochrome sodium sulfonate (AC-17) Carbazochrome sodium sulfonate (AC-17) (AC-17) is a capillary stabiliser and used for the research of haemorrhage.
- GC11419 Carbetocin oxytocin receptor agonist
- GC50450 Carboprost tromethamine Synthetic Prostaglandin F2α analog
- GC35610 Cariprazine hydrochloride An atypical antipsychotic
- GC46007 Cariprazine-d6 An internal standard for the quantification of cariprazine
-
GC68832
Carlumab
Carlumab (CNTO 888) is a highly-affinity humanized antibody against CCL2 (chemokine ligand 2). Carlumab can be used for cancer research, especially in prostate cancer.
- GC17864 CART (55-102) (human) CART with potent appetite-suppressing activity
- GC11131 CART (55-102) (rat) CART with potent appetite-suppressing activity
- GC14034 CART (62-76) (rat, human) CART (62-76) (rat, human) is a neuropeptide (62-76 residues of the CART peptide) with neurotransmitter-like effects.
- GC16395 Carteolol HCl Carteolol HCl (OPC-1085 hydrochloride) is a non-selective beta blocker used to treat glaucoma.
- GC14769 Carvedilol Potent β-adrenoceptor and α1-adrenoceptor antagonist
- GC25197 Carvedilol EP IMpurity E Carvedilol is a nonselective beta blocker/alpha-1 blocker and used in management of congestive heart failure (CHF).
- GC35613 Carvedilol phosphate hemihydrate Carvedilol phosphate hemihydrate (BM 14190 phosphate hemihydrate) is a non-selective β/α-1 blocker.
- GC64003 Carvedilol-d4
- GC16692 Casin GTPase Cdc42 inhibitor
- GC62888 Casopitant mesylate Casopitant mesylate (GW679769B) is a potent, selective, brain permeable and orally active neurokinin 1 (NK1) receptor antagonist.
- GC50293 CATPB FFA2 (GPR43) inverse agonist
- GC18318 CAY10441 CAY10441 is a potent and selective IP (prostacyclin) receptor antagonist.
- GC35620 CAY10471 Racemate CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist, with a Ki of 0.6 nM for hCRTH2, selective over human thromboxane A2 receptor TP (Ki, >10000 nM) or PGD2 receptor DP (Ki, 1200 nM).
- GC18678 CAY10595 The biological effects of prostaglandin D2 (PGD2) are transduced by at least two 7-transmembrane G protein-coupled receptors, designated DP1 and CRTH2/DP2.