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Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein

Products for  GPCR/G protein

  1. Cat.No. Product Name Information
  2. GC68435 Clazosentan Clazosentan Chemical Structure
  3. GC12778 Clenbuterol (hydrochloride) sympathomimetic β2-adrenoceptor agonist used as a bronchodilator in the treatment of pulmonary diseases Clenbuterol (hydrochloride) Chemical Structure
  4. GC68418 Clenbuterol-d9 Clenbuterol-d9 Chemical Structure
  5. GC62900 Clenproperol-D7 Clenproperol-D7 is the deuterium labeled Clenproperol. Clenproperol-D7 Chemical Structure
  6. GC31048 Clidinium bromide (Ro 2-3773) Clidinium bromide (Ro 2-3773) is a quaternary amine antimuscarinic agent. Clidinium bromide (Ro 2-3773) Chemical Structure
  7. GC11976 Clobetasol propionate Glucocorticoid receptor agonist Clobetasol propionate Chemical Structure
  8. GC39362 Clobetasone butyrate Clobetasone butyrate is a synthetic glucocorticoid and has topical anti-inflammatory activity especially in skin. Clobetasone butyrate Chemical Structure
  9. GC31037 Clocapramine (Clocarpramine) Clocapramine (Clocarpramine) Chemical Structure
  10. GC15107 Clomipramine HCl Clomipramine (Chlorimipramine) hydrochloride is a potent 5-HT reuptake blocker with the IC50 value of 1.5 nM. Clomipramine HCl Chemical Structure
  11. GC60717 Clonidine Clonidine is an alpha 2-adrenergic agonist. Clonidine Chemical Structure
  12. GC14032 Clonidine HCl Clonidine HCl is an agonist of α2-adrenoceptor and potent antihypertensive agent. Clonidine HCl Chemical Structure
  13. GC35710 Clopidogrel Clopidogrel is an orally active platelet inhibitor that targets P2Y12 receptor. Clopidogrel Chemical Structure
  14. GC15964 Clopidogrel hydrogen sulfate P2Y12 receptor antagonist Clopidogrel hydrogen sulfate Chemical Structure
  15. GC35711 Clopidogrel thiolactone Clopidogrel thiolactone is an active metabolites containing thiols resulting from thionolactone transformation of clopidogrel. Clopidogrel thiolactone Chemical Structure
  16. GC12949 Clorprenaline HCL Clorprenaline HCL is a β2-adrenergic receptor agonist that is implicated in bronchial expansion. Clorprenaline HCL Chemical Structure
  17. GC17760 Clozapine Clozapine (HF 1854) is an antipsychotic used for the research of schizophrenia. Clozapine Chemical Structure
  18. GC50193 Clozapine - d8 Clozapine - d8 (HF 1854-d8) is the deuterium labeled Clozapine. Clozapine - d8 Chemical Structure
  19. GC10822 Clozapine N-oxide (CNO)

    A metabolite of clozapine and muscarinic DREADD agonist

     Clozapine N-oxide (CNO) Chemical Structure
  20. GC63801 CM398 CM398 is a highly selective, orally active sigma-2 receptor ligand (Ki=0.43 nM), with high sigma-1/sigma-2 selectivity rato (1000-fold). CM398 Chemical Structure
  21. GC62347 CMC2.24 CMC2.24 (TRB-N0224), an orally active tricarbonylmethane agent, is effective against pancreatic tumor in mice by inhibiting Ras activation and its downstream effector ERK1/2 pathway. CMC2.24 Chemical Structure
  22. GC12627 Conivaptan HCl Conivaptan (hydrochloride) is a non-peptide antagonist of vasopressin receptor, with Ki values of 0.48 and 3.04 nM for rat liver V1A receptor and rat kidney V2 receptor respectively. Conivaptan HCl Chemical Structure
  23. GC18110 COR 170 inverse agonist of CB2 receptors COR 170 Chemical Structure
  24. GC50455 Cortagine Potent and selective CRF1 agonist Cortagine Chemical Structure
  25. GC12327 Corticosterone Corticosterone (17 deoxycortisol) is a glucocorticoid with oral activity and produced by adrenal cortex, which plays an important role in regulating the neuronal function of limbic system (including hippocampus, prefrontal cortex and amygdala). Corticosterone Chemical Structure
  26. GC60724 Corticotropin-releasing factor (human) (acetate) Corticotropin-releasing factor human acetate (Human CRF acetate) stimulates the synthesis and secretion of adrenocorticotropin in the anterior pituitary. Corticotropin-releasing factor (human) (acetate) Chemical Structure
  27. GC33839 Cortisone (17-Hydroxy-11-dehydrocorticosterone) Cortisone (17-Hydroxy-11-dehydrocorticosterone) Chemical Structure
  28. GC16772 Cortisone acetate Glucocorticoid receptor agonist Cortisone acetate Chemical Structure
  29. GC12835 Cortistatin 14 Cortistatin 14 (CST-14, human, rat), a neuropeptide with neuronal depressant and sleep modulating properties, can bind to all five cloned somatostatin receptors (SSTRs) and ghrelin receptor to exert its biological activities and co-exists with GABA within the cortex and hippocampus. Cortistatin 14 Chemical Structure
  30. GC35730 Cortistatin-14 TFA Cortistatin-14 (TFA), a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5). Cortistatin-14 TFA Chemical Structure
  31. GC10777 Cortistatin-8 ghrelin receptor antagonist Cortistatin-8 Chemical Structure
  32. GC39363 Cortodoxone Cortodoxone is a glucocorticoid steroid hormone that can be oxygenated to cortisol (Hydrocortisone). Cortodoxone Chemical Structure
  33. GC64090 Corydalmine Corydalmine (L-Corydalmine) inhibits spore germination of some plant pathogenic as well as saprophytic fungi. Corydalmine Chemical Structure
  34. GC39364 Cotadutide acetate Cotadutide (MEDI0382) acetate is a potent dual agonist of glucagon-like peptide-1 (GLP-1) and GCGR with EC50 values of 6.9 pM and 10.2 pM, respectively. Cotadutide acetate Chemical Structure
  35. GC47122 Coumaphos An organophosphate pesticide Coumaphos Chemical Structure
  36. GC50042 CP 122721 hydrochloride High affinity NK1 antagonist CP 122721 hydrochloride Chemical Structure
  37. GC11802 CP 135807 5-HT1D receptor agonist CP 135807 Chemical Structure
  38. GC12170 CP 154526 CRF1 receptor antagonist CP 154526 Chemical Structure
  39. GC31043 CP 316311

    CP 316311 is a potent and selective CRF1 receptor antagonist with an IC50 value of 6.8 nM.

     CP 316311 Chemical Structure
  40. GC30863 CP 376395 (CP-316311) CP 376395 (CP-316311) is a potent and selective Corticotropin releasing factor 1 (CRF1) receptor antagonist. CP 376395 (CP-316311) Chemical Structure
  41. GC10548 CP 376395 hydrochloride CRF1 receptor antagonist CP 376395 hydrochloride Chemical Structure
  42. GC10068 CP 93129 dihydrochloride 5-HT1B agonist, potent and highly selective CP 93129 dihydrochloride Chemical Structure
  43. GC16653 CP 94253 hydrochloride 5-HT1B agonist CP 94253 hydrochloride Chemical Structure
  44. GC32015 CP-105696 (Pfizer 105696) CP-105696 (Pfizer 105696) is a potent and selective Leukotriene B4 Receptor antagonist, with an IC50 of 8.42 nM. CP-105696 (Pfizer 105696) Chemical Structure
  45. GC17205 CP-945598 HCl CP-945598 HCl is a potent and selective cannabinoid receptor CB1 antagonist with Ki of 0.7 nM, exhibits 10,000-fold greater selectivity against human CB2 receptor. CP-945598 HCl Chemical Structure
  46. GC31923 CP-96486 CP-96486 is a potent and orally active leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor antagonist with Kis of 20 and 24 nM, respectively. CP-96486 Chemical Structure
  47. GC32734 CPI-444 (V81444) CPI-444 (V81444) (V81444) is a potent, orally active and selective adenosine A2A receptor (A2AR) antagonist, which induces antitumor responses. CPI-444 (V81444) Chemical Structure
  48. GC13426 CPPHA A positive allosteric modulator of the mGluR5 CPPHA Chemical Structure
  49. GC14137 CRF (6-33) CRF (6-33) is a CRF binding protein (CRF-BP) ligand inhibitor. CRF (6-33) Chemical Structure
  50. GC15737 CRF (human, rat) Corticotropin-releasing factor human (Human CRF) stimulates the synthesis and secretion of adrenocorticotropin in the anterior pituitary. CRF (human, rat) Chemical Structure
  51. GC35748 CRF, bovine CRF, bovine is a potent agonist of CRF receptor, and displaces [125I-Tyr]ovine CRF with a Ki of 3.52 nM. CRF, bovine Chemical Structure
  52. GC34542 CRF, bovine TFA CRF, bovine (TFA) is a potent agonist of CRF receptor, and displaces [125I-Tyr]ovine CRF with a Ki of 3.52 nM. CRF, bovine TFA Chemical Structure
  53. GC18099 CRSP-1 Endogenous central calcitonin (CT) receptor agonist CRSP-1 Chemical Structure
  54. GC31903 CRTh2 antagonist 1 CRTh2 antagonist 1 is a CRTh2 antagonist with an IC50 of 89 nM. CRTh2 antagonist 1 Chemical Structure
  55. GC31998 CRTH2-IN-1 (Ramatroban analog) CRTH2-IN-1 (Ramatroban analog) (Ramatroban analog) is a selective prostaglandin D2 receptor DP2 (CRTH2) antagonist with an IC50 of 6 nM in a human DP2 binding assay. CRTH2-IN-1 (Ramatroban analog) Chemical Structure
  56. GC13966 CS 2100 S1P1 agonist CS 2100 Chemical Structure
  57. GC35751 CS-003 Free base CS-003 Free base (CS-003), a triple tachykinin receptor antagonist, shows high affinities for human (Neurokinin) NK1, NK2 and NK3 receptors with Ki values of 2.3 nM, 0.54 nM and 0.74 nM, respectively. CS-003 Free base Chemical Structure
  58. GC65450 CT1812 CT1812 (Sigma-2 receptor antagonist 1) is a sigma-2 (σ-2) receptor antagonist. CT1812 Chemical Structure
  59. GC13360 CTCE 9908 CXCR4 antagonist CTCE 9908 Chemical Structure
  60. GC16619 CTEP (RO4956371) CTEP (RO4956371) (RO 4956371) is a novel, long-acting, orally bioavailable allosteric antagonist ofmGlu5receptor withIC50of 2.2 nM, and shows > 1000-fold selectivity over other mGlu receptors. CTEP (RO4956371) Chemical Structure
  61. GC68909 Cudarolimab

    Cudarolimab (IBI101) is a fully human anti-OX40 (CD134, a co-stimulatory molecule expressed by activated immune cells) antibody. Cudarolimab inhibits the binding of OX40 to its ligand OX40L. Cudarolimab has anti-tumor activity and can be used in cancer-related research.

     Cudarolimab Chemical Structure
  62. GC33697 Cutamesine (SA4503) Cutamesine (SA4503) (SA4503; AGY-94806) is a selective sigma 1 receptor(σ1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4±1.9 nM); 100-fold less affinity for the sigma 2 receptor. Cutamesine (SA4503) Chemical Structure
  63. GC14706 CV 1808 Adenosine A2 receptor agonist CV 1808 Chemical Structure
  64. GC65908 CXCR2 antagonist 2 CXCR2 antagonist 2 is a potent CXCR2 antagonist for cancer immunotherapy with an IC50 value of 95 nM. CXCR2 antagonist 2 Chemical Structure
  65. GC31754 CXCR2-IN-1 CXCR2-IN-1 is a central nervous system penetrant CXCR2 antagonist with a pIC50 of 9.3. CXCR2-IN-1 Chemical Structure
  66. GC62475 CXCR2-IN-2 CXCR2-IN-2 is a selective, brain penetrant, and orally bioavailable CXCR2 antagonist (IC50=5.2 nM/1 nM in β-arrestin assay/CXCR2 Tango assay, respectively). CXCR2-IN-2 Chemical Structure
  67. GC63411 CXCR7 antagonist-1

    CXCR7 antagonist-1 is a CXCR7 antagonist that inhibits the binding of the SDF-1 chemokine (also known as the CXCL12 chemokine) or I-TAC (also known as CXCL11) to the chemokine receptor CXCR7.

     CXCR7 antagonist-1 Chemical Structure
  68. GC65476 CXCR7 antagonist-1 hydrochloride CXCR7 antagonist-1 hydrochloride is a CXCR7 antagonist that inhibits the binding of the SDF-1 chemokine (also known as the CXCL12 chemokine) or I-TAC (also known as CXCL11) to the chemokine receptor CXCR7. CXCR7 antagonist-1 hydrochloride Chemical Structure
  69. GC35763 CXCR7 modulator 1 CXCR7 modulator 1 (compound 25) is a potent and orally bioavailable peptoid hybrid CXCR7 modulator, with a Ki of 9 nM. CXCR7 modulator 1 Chemical Structure
  70. GC34339 CXCR7 modulator 2 CXCR7 modulator 2 is a modulator of C-X-C Chemokine Receptor Type 7 (CXCR7), with a Ki of 13 nM. CXCR7 modulator 2 Chemical Structure
  71. GC38760 Cyamemazine Cyamemazine is a neuroleptic agent that contains the phenothiazine chromophore. Cyamemazine Chemical Structure
  72. GC43341 Cyclic GMP

    Guanosine 3',5'-cyclic monophosphate (cyclic GMP or cGMP) is a second messenger that is biosynthesized from GTP by guanylate cyclases.

     Cyclic GMP Chemical Structure
  73. GC10743 Cyclobenzaprine HCl Cyclobenzaprine HCl (MK130 hydrochloride) is a skeletal muscle relaxant and a central nervous system (CNS) depressant. Cyclobenzaprine HCl Chemical Structure
  74. GC31209 Cyclodrine hydrochloride Cyclodrine hydrochloride is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist. Cyclodrine hydrochloride Chemical Structure
  75. GC43347 Cyclopentolate (hydrochloride) Cyclopentolate is an antagonist of muscarinic acetylcholine receptors (Kis = 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively). Cyclopentolate (hydrochloride) Chemical Structure
  76. GC15495 Cyclosomatostatin somatostatin receptor antagonist Cyclosomatostatin Chemical Structure
  77. GC15319 Cyclosporin H

    Selective and competitive formyl peptide receptor antagonist

     Cyclosporin H Chemical Structure
  78. GC10728 CYM 50260 S1P4 agonist CYM 50260 Chemical Structure
  79. GC15903 CYM 50308 S1P4 agonist CYM 50308 Chemical Structure
  80. GC14350 CYM 50358 hydrochloride S1P4 antagonist CYM 50358 hydrochloride Chemical Structure
  81. GC18138 CYM 50769 neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist CYM 50769 Chemical Structure
  82. GC16567 CYM 5442 hydrochloride S1P1 agonist, potent and selective CYM 5442 hydrochloride Chemical Structure
  83. GC15765 CYM 5520

    noncompetitive allosteric agonist of S1P2

     CYM 5520 Chemical Structure
  84. GC16946 CYM 5541 sphingosine-1-phosphate receptor 3 (S1P3) allosteric agonist CYM 5541 Chemical Structure
  85. GC17307 CYM 9484 neuropeptide Y (NPY) Y2 receptor antagonist CYM 9484 Chemical Structure
  86. GC63345 CYM50358 CYM50358 is a potent and selective S1PR4 antagonist, with an IC50 of 25 nM. CYM50358 Chemical Structure
  87. GC14747 CYN 154806 somatostatin sst2 receptor antagonist CYN 154806 Chemical Structure
  88. GC35787 CYN 154806 TFA CYN 154806 TFA, a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively. CYN 154806 TFA Chemical Structure
  89. GC65565 Cyproheptadine Cyproheptadine is a potent and orally active 5-HT2A receptor antagonist, with antidepressant and antiserotonergic effects. Cyproheptadine Chemical Structure
  90. GC43353 Cyproheptadine (hydrochloride hydrate) Cyproheptadine (hydrochloride hydrate) is an antihistamine and is an antagonist of serotonin and histamine2. Cyproheptadine (hydrochloride hydrate) Chemical Structure
  91. GC10698 Cyproheptadine hydrochloride serotonin and histamine antagonist as well as antimuscarinic reagent Cyproheptadine hydrochloride Chemical Structure
  92. GC30665 D2343 D2343 is a β2-adrenoceptor agonist and also is an α1- adrenoceptor inhibitor. D2343 Chemical Structure
  93. GC60737 D3-βArr D3-βArr Chemical Structure
  94. GC38762 Dabuzalgron Dabuzalgron (Ro 115-1240) is an orally active and selective α-1A adrenergic receptor agonist for the treatment of urinary incontinence. Dabuzalgron Chemical Structure
  95. GC31844 Dagrocorat (PF-00251802) Dagrocorat (PF-00251802) (PF-00251802) is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat (PF-00251802) Chemical Structure
  96. GC63872 Dagrocorat hydrochloride Dagrocorat (PF-00251802) hydrochloride is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat hydrochloride Chemical Structure
  97. GC38763 Daltroban Daltroban (BM-13505) is a selective and specific thromboxane A2 (TXA2) receptor antagonist. Daltroban Chemical Structure
  98. GC65550 Danavorexton Danavorexton is an orexin receptor agonist. Danavorexton Chemical Structure
  99. GC19116 Danirixin Danirixin is a selective, and reversible CXCR2 antagonist, with IC50 of 12.5 nM for CXCL8. Danirixin Chemical Structure
  100. GC30188 Dapiprazole hydrochloride An α-adrenergic receptor antagonist Dapiprazole hydrochloride Chemical Structure
  101. GC17061 Dapoxetine HCl Selective serotonin reuptake inhibitor Dapoxetine HCl Chemical Structure

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