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Products for Others
- Cat.No. Product Name Information
- GC49473 ARA 290 (acetate) A derivative of EPO
- GC39340 Arachidonyl alcohol Arachidonyl alcohol is a long-chain primary fatty alcohol.
- GC19435 Aramchol Aramchol, also known as arachidyl amido cholanoic acid, is a conjugate of arachidic acid and cholic acid .
- GC48997 Argipressin (acetate) A peptide hormone with vasoconstrictive and antidiuretic activities
- GC35389 Aristolochic acid B An alkaloid with mutagenic activity
- GC35392 Aristolone Aristolone is a sesquiterpene isolated from Aristolochia debilis.
- GC17225 ARL 67156 trisodium salt ARL67156 (FPL 67156) trisodium is a selective ecto-ATPase inhibitor.
- GC62848 ARN 077 (enantiomer) ARN 077 enantiomer (19) is the less active enantiomer of ARN 077, with an IC50 of 3.53 μM for rat NAAA.
- GC31913 ARN 077 (URB913) ARN 077 (URB913) is a potent and selective N-acylethanolamine acid amidase (NAAA) inhibitor with an IC50 of 7 nM for human NAAA.
- GC41215 ARN14686 ARN14686 is an activity-based affinity probe for the detection of N-acylethanolamine acid amidase (NAAA) using click chemistry.
- GC63794 ARN19702 ARN19702 is a selective, orally active, reversible, and brain-penetrant N-acylethanolamine acid amidase (NAAA) inhibitor with an IC50 of 230 nM for human NAAA.
- GC18448 ARN272 ARN272 is an anandamide transport inhibitor.
- GC45386 ARN726 ARN726 is a potent NAAA (N-acylethanolamine acid amidase) inhibitor with an IC50 of 0.073 μM.
- GC32668 Arrhythmias-Targeting Compound 1 Arrhythmias-Targeting Compound 1 is used in the research of arrhythmias, extracted from patent WO 2001028992 A2.
- GC32669 Arrhythmic-Targeting Compound 1 Arrhythmic-Targeting Compound 1 is used for the research of arrhythmic disease, with nitrogen-containing spirocycles.
- GC64426 ART812 ART812 is an orally active DNA polymerase Polθ inhibitor with an IC50 value of 7.6 nM. ART812 has an IC50 value of 240 nM for cell based microhomology-mediated end joining (MMEJ).
- GC10889 Artesunate Derivative of the natural product artemisinin
- GC13404 Articaine HCl Articaine HCl (Hoe-045) is an amide anaesthetic containing an ester group, reversibly binding to the α-subunit of the voltage-gated sodium channels within the inner cavity of the nerve, can provide effective pain relief.
- GC17659 AS 101 AS 101 (AS101), an immunomodulatory tellurium compound, is a potent IL-1β inhibitor.
- GC64909 AS057278 AS057278 is a potent, selective, orally active and blood-brain barrier (BBB) penetrant non-peptidic D-amino acid oxidase (DAAO) inhibitor with an IC50 value of 0.91 μM and EC50 of 2.2-3.95 μM.
- GC12070 Ascorbic acid An electron donor
- GC35402 Ascr#2 Ascr#2 is an ascaroside isolated from Caenorhabditis elegans, potently promotes dauer formation, and also acts as a potent male attractant combined with ascr#3 at low concentration.
- GC35403 Ascr#3 Ascr#3 is an ascaroside isolated from Caenorhabditis elegans, acts a potent male attractant, and also promotes dauer formation combined with ascr#2 at low concentration.
- GC35404 Ascr#5 Ascr#5 is a highly conserved ascaroside isolated from Caenorhabditis elegans.
- GC35405 Ascr#8 Ascr#8 is an dauer-inducing ascaroside isolated from Caenorhabditis elegans, synergizes with ascr#2 and ascr#3, and strongly enhances male attraction.
- GC32936 ASP-9521 An inhibitor of 17β-HSD5/AKR1C3
- GC30004 Asparagusic acid Asparagusic acid is a sulfur-containing flavor component produced by asparagus plants, with anti-parasitic effect.
- GC12862 Aspartame non-saccharide sweetener
- GC35410 Aspartyl-alanyl-diketopiperazine Aspartyl-alanyl-diketopiperazine (DA-DKP) is an immunomodulatory molecule generated by cleavage and cyclization from the N-terminus of human albumin and can modulate the inflammatory immune response through a molecular pathway implicated in T- lymphocyte anergy.
- GC33886 Aspirin Aluminum (Aluminum diacetylsalicylate) Aspirin Aluminum (Aluminum diacetylsalicylate) is a novel intermolecular compound which can inhibit gastrointestinal mucosal disorders induced by NSAIDs (non-steroidal anti-inflammatory agents) extracted from patent WO 2010064441 A1.
- GC32014 Asthma relating compound 1 Asthma relating compound 1 is an anti-asthmatic agent candidate extracted from patent EP0295656A1.
- GC62852 Astragenol Astragenol is an intermediate used for Astragenol derivative synthesis.
- GC12537 ATB-337 ATB-337 is a hybrid molecule of an H2S donor and the NSAID diclofenac.
- GC16245 ATB-343 hybrid molecule of an H2S donor and the NSAID indomethacin
- GC32200 ATB107 ATB107 is a novel and potent inhibitor of indole-3-glycerol phosphate synthase (IGPS) with a KD of 3 μM.
- GC15770 Atglistatin ATGL inhibitor, potent and selective
- GC35417 Athidathion Athidathion(GS-13006) is an organophosphate insecticide.
- GC18537 ATN-224 ATN-224 is a choline salt of tetrathiomolybdate and an inhibitor of superoxide dismutase 1 (SOD1; IC50s = 2.91 and 3.51 uM in human and mouse blood cells, respectively, in vitro).
- GC10274 Atomoxetine HCl Atomoxetine HCl is a potent and selective noradrenalin re-uptake inhibitor (Ki values are 5, 77 and 1451 nM for inhibition of radioligand binding to human NET, SERT and DAT respectively).
- GC63818 Atorvastatin acetonide tert-butyl ester Atorvastatin acetonide tert-butyl ester is a useful pharmaceutical intermediate in the preparation of Atorvastatin salts.
- GC66040 ATPase-IN-2 ATPase-IN-2 is an ATPase inhibitor with an IC50 value of 0.9 μM. ATPase-IN-2 inhibits C. difficile toxin B (TcdB) glycohydrolase activity with an AC50 value of 30.91 μM. ATPase-IN-2 can be used for the research of ATP-related.
- GC42869 Atpenin A5 Mitochondrial complex II (succinate dehydrogenase or succinate:ubiquinone oxidoreductase) is a functional member of the Krebs cycle and the aerobic respiratory chain that couples the oxidation of succinate to fumarate with the reduction of quinone to quinol.
- GC60059 Atrazine Atrazine is principally used for control of certain annual broadleaf and grass weeds.
- GC34155 Atrimustine (Bestrabucil) Atrimustine (Bestrabucil) is a conjugate of chlorambucil and β-estradiol benzoate with the antitumor activity.
- GC34219 ATWLPPR Peptide TFA ATWLPPR Peptide TFA, a heptapeptide, acts as a selective neuropilin-1 inhibitor, inhibits VEGF165 binding to NRP-1, used in the research of angiogenesis.
- GC65532 ATX-002 ATX-002 is a property-tunable lipid for RNA drug delivery.
- GC64272 AU-16235 AU-16235 is an inactive epimer of AU-15330. AU-16235 has no effect on cancer cell survival and growth
- GC31568 AU-224 AU-224 is a benzamide derivative used as a promising gastrointestinal prokinetic agent without significant side effects.
- GC35431 Aurothioglucose Aurothioglucose (Gold thioglucose) is a well known active-site inhibitor of TrxR1, inhibited TrxR1 activity in HeLa cell cytosol but had no effect on the viability of the cells.
- GC30028 Auxinole Auxinole is a potent auxin antagonist of TIR1/AFB receptors, binding TIR1 to block the formation of the TIR1-IAA-Aux/IAA complex and so inhibits auxin-responsive gene expression.
- GC42877 AUY954 AUY954 is an orally bioavailable and selective agonist of the sphingosine-1-phosphate receptor 1 (S1P1; EC50 = 1.2 nM for stimulating GTPγS binding to S1P1 in CHO cells).
- GC64329 Avasopasem manganese Avasopasem manganese (GC4419; M-40419) is a potent superoxide dismutase mimetic that rapidly and specifically converts O2*- to hydrogen peroxide (H2O2), arresting the initiation of this cascade.
- GC31627 AVE5688 AVE5688 is an inhibitor of glycogen phosphorylase (GP), with IC50s of 430 nM and 915 nM and Kds of 170 nM and 530 nM for rabbit muscle glycogen phosphorylase (rmGPb and rmGPa, respectively); AVE5688 can be used for the research of type 2 diabetes.
- GC19045 AVN-944 AVN-944(VX-944) is a selective, noncompetitive inhibitor of the enzyme directed against human IMPDH with Ki of 6-10 nM for IMPDH1/IMPDH2.
- GC14614 Avobenzone topical, broad range UV protector
- GC30139 Avoralstat (BCX4161) Avoralstat (BCX4161) (BCX4161), a potent and orally active plasma kallikrein (PKK) inhibitor, is used for hereditary angioedema research.
- GC63301 AWL-II-38.3 AWL-II-38.3 is a potent ephrin-A receptor (EphA3) kinase inhibitor. AWL-II-38.3 does not exhibit significant cellular activity against Src-family kinases nor against b-raf.
- GC65496 AXKO-0046 AXKO-0046 is an indole derivative and small-molecule LDHB selective inhibitor.
- GC64853 Axomadol Axomadol (EN3324) is a centrally active analgesic agent with opioid agonistic properties and inhibitory effects on the reuptake of monoamines.
- GC12429 AY 9944 dihydrochloride AY 9944 dihydrochloride is a specific cholesterol biosynthesis inhibitor.
- GC34479 AZ PFKFB3 26 AZ PFKFB3 26 is a potent and selective inhibitor of the metabolic kinase PFKFB3 with an IC50 of 23 nM. AZ PFKFB3 26 inhibits PFKFB1 and PFKFB2 with IC50s of 2.06 and 0.384 μM, respectively.
- GC50250 AZ PFKFB3 67 Potent and selective PFKFB3 inhibitor
- GC62858 AZ-PFKFB3-67 quarterhydrate AZ-PFKFB3-67 quarterhydrate is potent and selective metabolic kinase PFKFB3 inhibitor, with IC50s of 11, 159 and 1130 nM for PFKFB3, PFKFB2 and PFKFB1 respectively.
- GC16119 Azacyclonol tranquilizer,antipsychotic
- GC14874 Azaserine tumor-inhibiting antibiotic
- GC31601 AZD 4017 AZD 4017 is a potent, selective 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) inhibitor, with an IC50 of 7 nM.
- GC63551 AZD-CO-Ph-PEG4-Ph-CO-AZD AZD-CO-Ph-PEG4-Ph-CO-AZD is a bis-β-lactam linker can be used for antibody-siRNA conjugate synthesis.
- GC35449 AZD8329 AZD8329 is a potent 11β-Hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor with an IC50 of 9 nM for human 11β-HSD1, displays excellent selectivity versus 11β-HSD2, 17β-HSD1 and 17β-HSD3.
- GC30508 Azelaprag
- GC34337 AzKTB AzKTB is a capture reagent which bears a short trypsin-cleavable peptide sequence between the azide module and the TAMRA/PEG-biotin labels.
- GC30634 Azobenzene Azobenzene can be used as an optical trigger for the design and synthesis of a large variety of photoresponsive systems.
- GC14184 Azomycin antimicrobial antibiotic
- GC19445 Azoxymethane Azoxymethane, as a colon carcinogen, can lead to the formation of DNA adducts. Azoxymethane (AOM) causes O(6)-methylguanine adduct formation which leads to G-->A transitions. .
- GP10125 b-Casomorphin (1-3)
- GC60618 B7/CD28 interaction inhibitor 1 B7/CD28 interaction inhibitor 1 (copmound 6b) is a potent B7.1-CD28 interaction inhibitor with an IC50 of 50 nM.
- GC42894 Baccatin III Baccatin III is a polycyclic diterpene originally isolated from the yew tree (Taxus) that is a precursor of paclitaxel.
- GC64861 Bafrekalant Bafrekalant is a diazabicyclic substituted imidazo[l,2-a]pyrimidine-derivative.
- GC52344 Bak BH3 (72-87) (human) (trifluoroacetate salt) A Bak-derived peptide
- GC61860 Baldrinal Baldrinal is derived from the extracts of valerian rhizomes and roots, inhibits autonomic activity, and has anti-inflammatory effects.
-
GC19056
BAM 15
BAM 15 is a novel mitochondrial protonophore uncoupler.
- GC14668 BAMB-4 Inositol-1,4,5-trisphosphate-3-kinase A (ITPKA) inhibitor
- GC13517 BAPTA-AM BAPTA-AM is a well-known membrane-permeable Ca2+ chelator, to prevent cell injury by allaying the intracellular calcium overload
- GC38351 Barbadin Barbadin is a novel and selective β-arrestin/β2-adaptin interaction inhibitor, has IC50 values of 19.1?μM for β-arrestin1 and 15.6?μM for β-arrestin2.
- GC67537 Basic Brown 1 Basic Brown 1 is a diazo dyes.
- GC65952 BAY-091 BAY-091 is a novel potent and highly selective inhibitor of the kinase PIP4K2A.
- GC32824 BAY-1816032 BAY-1816032 is a potent and oral available BUB1 (budding uninhibited by benzimidazoles 1) kinase inhibitor with an IC50 of 7 nM.
- GC62861 BAY-298 BAY-298 is an orally active and selective luteinizing hormone receptor (LH-R) antagonist with IC50s of 96 nM, 23 nM and 78 nM for hLH (human LH) and rLH (rat LH) and cLH (cynomolgus monkey LH), respectively.
- GC34164 BAY-320 BAY-320 is a Bub1 inhibitor, with an IC50 of 680 nM for human Bub1 in the presence of 2 mM ATP.
- GC33236 BAY-524 BAY-524 is a potent Bub1 kinase inhibitor. BAY-524 inhibits the recombinant catalytic domain of human Bub1 with an IC50 of 450 nM. BAY-524 can be used for the research of anti-cancer in combination with other agents.
- GC30619 BAY-677 BAY-677 is an inactive control for BAY-678.
- GC35477 BAY-826 BAY-826 is a selective and potent TIE-2 inhibitor with a Kd of 1.6 nM, respectively.
- GC31484 BAY-850 BAY-850 is a potent and isoform selective ATPase family AAA domain-containing protein 2 (ATAD2) inhibitor, with an IC50 of 166 nM.
- GC19061 BAY-876 BAY-876 is the first highly selective GLUT1 inhibitor with IC50 of 0.002 uM.
- GC66409 BAY-888 BAY-888 exhibits IC50 value of 1.5 nM and 5.5 nM towards CSNK1A1 and CSNK1D, respectively.
- GC61746 BAY-899 BAY-899 is an orally active and selective luteinizing hormone receptor (LH-R) antagonist with IC50s of 185 nM and 46nM for hLH (human LH) and rLH (rat LH), respectively.
- GC64132 BCAT-IN-1 BCAT-IN-1 is a potent, selective and orally active inhibitor of BCATm, with a pIC50 of 7.3.
- GC62862 BCAT-IN-2 BCAT-IN-2 is a potent, selective and orally active inhibitor of mitochondrial branched-chain aminotransferase (BCATm), with a pIC50 of 7.3.
- GC65257 BCL6-IN-6 BCL6-IN-6 is a potent inhibitor of transcriptional repressor B-cell lymphoma 6 (BCL6). BCL6-IN-6 significantly blocks the interaction of BCL6 with its corepressors and reactivates BCL6 target genes in a dose-dependent manner. BCL6-IN-6 has the potential for the research of diffuse large B-cell lymphoma (DLBCL).
- GC61612 BDP-13176 BDP-13176 is a potent fascin 1 inhibitor, with a Kd of 90 nM and an IC50 of 240 nM. BDP-13176 has potential as an anti-metastatic agent.
- GC50173 BDY 650-X, SE Red BDY (BODIPY® or boron-dipyrromethene) fluorescent dye for the labeling of amines; supplied as NHS ester